Publications by authors named "Sandeep Ghorpade"

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Optimization of 2,8-Diaryl-1,5-naphthyridines as Phosphatidylinositol 4-Kinase Inhibitors with Improved ADME Profiles and In Vivo Efficacy.
Godwin A Dziwornu, Donald Seanego, Stephen Fienberg, Venkata S Sypu, Nicolaas Salomane, Sandeep R Ghorpade

J Med Chem· October 2025

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Novel Inhibitors of Phosphatidylinositol 4-kinase IIIβ with Low Propensity for Resistance: Life Cycle Stage Activity and Efficacy in a Humanized Mouse Malaria Infection Model.
Godwin A Dziwornu, Mmakwena M Mmonwa, Dina Coertzen, Liezl Krugmann, Nicolaas Salomane, Sandeep R Ghorpade

J Med Chem· August 2025

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2,8-Disubstituted-1,5-naphthyridines as Dual Inhibitors of Phosphatidylinositol-4-kinase and Hemozoin Formation with Efficacy.
Godwin Akpeko Dziwornu, Donald Seanego, Stephen Fienberg, Monica Clements, Jasmin Ferreira, Sandeep R Ghorpade

J Med Chem· July 2024

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Recent developments of imidazo[1,2-]pyridine analogues as antituberculosis agents.
Sauvik Samanta, Sumit Kumar, Eswar K Aratikatla, Sandeep R Ghorpade, Vinayak Singh

RSC Med Chem· April 2023

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1,3-Diarylpyrazolyl-acylsulfonamides Target HadAB/BC Complex in .
Vinayak Singh, Anna E Grzegorzewicz, Stephen Fienberg, Rudolf Müller, Lutete Peguy Khonde, Sandeep R Ghorpade

ACS Infect Dis· November 2022

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Spiropyrimidinetrione DNA Gyrase Inhibitors with Potent and Selective Antituberculosis Activity.
Preshendren Govender, Rudolf Müller, Kawaljit Singh, Virsinha Reddy, Charles J Eyermann, Sandeep R Ghorpade

J Med Chem· May 2022

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Spiropyrimidinetriones: a Class of DNA Gyrase Inhibitors with Activity against Mycobacterium tuberculosis and without Cross-Resistance to Fluoroquinolones.
Gregory S Basarab, Sandeep Ghorpade, Liezl Gibhard, Rudolf Mueller, Mathew Njoroge

Antimicrob Agents Chemother· April 2022

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1,3-Diarylpyrazolyl-acylsulfonamides as Potent Anti-tuberculosis Agents Targeting Cell Wall Biosynthesis in .
Lutete Peguy Khonde, Rudolf Müller, Grant A Boyle, Virsinha Reddy, Aloysius T Nchinda, Sandeep R Ghorpade

J Med Chem· September 2021

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Antitubercular 2-Pyrazolylpyrimidinones: Structure-Activity Relationship and Mode-of-Action Studies.
Candice Soares de Melo, Vinayak Singh, Alissa Myrick, Sandile B Simelane, Dale Taylor, Sandeep R Ghorpade

J Med Chem· January 2021

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Novel Antitubercular 6-Dialkylaminopyrimidine Carboxamides from Phenotypic Whole-Cell High Throughput Screening of a SoftFocus Library: Structure-Activity Relationship and Target Identification Studies.
Colin R Wilson, Richard K Gessner, Atica Moosa, Ronnett Seldon, Digby F Warner, Sandeep R Ghorpade

J Med Chem· December 2017

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Whole cell screen based identification of spiropiperidines with potent antitubercular properties.
Subramanyam J Tantry, Giulia Degiacomi, Sreevalli Sharma, Lalit Kumar Jena, Ashwini Narayan, Sandeep R Ghorpade

Bioorg Med Chem Lett· August 2015

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2-Phenylindole and Arylsulphonamide: Novel Scaffolds Bactericidal against Mycobacterium tuberculosis.
Maruti Naik, Sandeep Ghorpade, Lalit Kumar Jena, Gopinath Gorai, Ashwini Narayan

ACS Med Chem Lett· September 2014

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4-aminoquinolone piperidine amides: noncovalent inhibitors of DprE1 with long residence time and potent antimycobacterial activity.
Maruti Naik, Vaishali Humnabadkar, Subramanyam J Tantry, Manoranjan Panda, Ashwini Narayan, Sandeep R Ghorpade

J Med Chem· June 2014

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Thiazolopyridone ureas as DNA gyrase B inhibitors: optimization of antitubercular activity and efficacy.
Ramesh R Kale, Manoj G Kale, David Waterson, Anandkumar Raichurkar, Shahul P Hameed, Sandeep R Ghorpade

Bioorg Med Chem Lett· February 2014

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Thiazolopyridine ureas as novel antitubercular agents acting through inhibition of DNA Gyrase B.
Manoj G Kale, Anandkumar Raichurkar, Shahul Hameed P, David Waterson, David McKinney, Sandeep R Ghorpade

J Med Chem· November 2013

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Binding of matrix metalloproteinase inhibitors to extracellular matrix: 3D-QSAR analysis.
Yufen Zhang, Viera Lukacova, Vladimir Bartus, Xiaoping Nie, Guorong Sun, Sandeep R Ghorpade

Chem Biol Drug Des· October 2008

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Enantioselective synthesis of alpha,beta-disubstituted-beta-amino acids.
Mukund P Sibi, Prabagaran Narayanasamy, Sandeep G Ghorpade, Craig P Jasperse

J Am Chem Soc· October 2003

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A convenient method for the conversion of N-acyloxazolidinones to hydroxamic acids.
Mukund P Sibi, Hikaru Hasegawa, Sandeep R Ghorpade

Org Lett· October 2002

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