Publications by authors named "Sandeep K Talapatra"

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Tetrazole-containing naphthalene bis-sulfonamide Keap1-Nrf2 interaction inhibitors with unexpected binding modes.
Nikolaos D Georgakopoulos, Sandeep K Talapatra, Sharadha Dayalan Naidu, Dina Dikovskaya, Maureen Higgins

Redox Biol· December 2025

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Structural and Molecular Insight into the PWWP1 Domain of NSD2 from the Discovery of Novel Binders Via DNA-Encoded Library Screening.
Gavin W Collie, Bryony Ackroyd, Catriona Corbishley, Daniel H O'Donovan, Alex Edwards, Sandeep K Talapatra

ACS Med Chem Lett· September 2025

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Is the Fate of Clinical Candidate Arry-520 Already Sealed? Predicting Resistance in Eg5-Inhibitor Complexes.
Rose-Laure Indorato, Sandeep K Talapatra, Fangzhu Lin, Shozeb Haider, Simon P Mackay

Mol Cancer Ther· December 2019

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The depolymerase activity of MCAK shows a graded response to Aurora B kinase phosphorylation through allosteric regulation.
Toni McHugh, Juan Zou, Vladimir A Volkov, Aurélie Bertin, Sandeep K Talapatra

J Cell Sci· January 2019

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Development and validation of RdRp Screen, a crystallization screen for viral RNA-dependent RNA polymerases.
Federica Riccio, Sandeep K Talapatra, Sally Oxenford, Richard Angell, Michela Mazzon

Biol Open· January 2019

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Modified Peptide Inhibitors of the Keap1-Nrf2 Protein-Protein Interaction Incorporating Unnatural Amino Acids.
Nikolaos D Georgakopoulos, Sandeep K Talapatra, Jemma Gatliff, Frank Kozielski, Geoff Wells

Chembiochem· September 2018

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Crystal structure of the Eg5 - K858 complex and implications for structure-based design of thiadiazole-containing inhibitors.
Sandeep K Talapatra, Chuin Lean Tham, Paolo Guglielmi, Roberto Cirilli, Balakumar Chandrasekaran

Eur J Med Chem· August 2018

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The structure of the binary methyltransferase-SAH complex from Zika virus reveals a novel conformation for the mechanism of mRNA capping.
Chatrin Chatrin, Sandeep K Talapatra, Bruno Canard, Frank Kozielski

Oncotarget· January 2018

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Depsidones from Lichens as Natural Product Inhibitors of M-Phase Phosphoprotein 1, a Human Kinesin Required for Cytokinesis.
Sandeep K Talapatra, Oliver Rath, Eddie Clayton, Sophie Tomasi, Frank Kozielski

J Nat Prod· June 2016

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New MKLP-2 inhibitors in the paprotrain series: Design, synthesis and biological evaluations.
Christophe Labrière, Sandeep K Talapatra, Sylviane Thoret, Cécile Bougeret, Frank Kozielski

Bioorg Med Chem· February 2016

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The C-terminal region of the motor protein MCAK controls its structure and activity through a conformational switch.
Sandeep K Talapatra, Bethany Harker, Julie P I Welburn

Elife· April 2015

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Analysis of the human cofilin 1 structure reveals conformational changes required for actin binding.
Marta Klejnot, Mads Gabrielsen, Jenifer Cameron, Andrzej Mleczak, Sandeep K Talapatra

Acta Crystallogr D Biol Crystallogr· September 2013

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Mitotic kinesin Eg5 overcomes inhibition to the phase I/II clinical candidate SB743921 by an allosteric resistance mechanism.
Sandeep K Talapatra, Nahoum G Anthony, Simon P Mackay, Frank Kozielski

J Med Chem· August 2013

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Optimized S-trityl-L-cysteine-based inhibitors of kinesin spindle protein with potent in vivo antitumor activity in lung cancer xenograft models.
James A D Good, Fang Wang, Oliver Rath, Hung Yi Kristal Kaan, Sandeep K Talapatra

J Med Chem· March 2013

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Structural insights into a unique inhibitor binding pocket in kinesin spindle protein.
Venkatasubramanian Ulaganathan, Sandeep K Talapatra, Oliver Rath, Andrew Pannifer, David D Hackney

J Am Chem Soc· February 2013

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Indolobenzazepin-7-ones and 6-, 8-, and 9-membered ring derivatives as tubulin polymerization inhibitors: synthesis and structure--activity relationship studies.
Aurélien Putey, Florence Popowycz, Quoc-Tuan Do, Philippe Bernard, Sandeep K Talapatra

J Med Chem· October 2009

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