Publications by authors named "Stefania Colarusso"

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SAR evolution towards potent C-terminal carboxamide peptide inhibitors of Zika virus NS2B-NS3 protease.
Stefania Colarusso, Federica Ferrigno, Simona Ponzi, Francesca Pavone, Immacolata Conte

Bioorg Med Chem· March 2022

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Guiding Chemically Synthesized Peptide Drug Lead Optimization by Derisking Mast Cell Degranulation-Related Toxicities of a NaV1.7 Peptide Inhibitor.
Pierre Morissette, Nianyu Li, Jeanine E Ballard, Marissa Vavrek, Gregory L Adams, Stefania Colarusso

Toxicol Sci· January 2022

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Development of ProTx-II Analogues as Highly Selective Peptide Blockers of Na1.7 for the Treatment of Pain.
Gregory L Adams, Parul S Pall, Steven M Grauer, Xiaoping Zhou, Jeanine E Ballard, Stefania Colarusso

J Med Chem· January 2022

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Optimization of linear and cyclic peptide inhibitors of KEAP1-NRF2 protein-protein interaction.
Stefania Colarusso, Daniele De Simone, Tommaso Frattarelli, Matteo Andreini, Mauro Cerretani

Bioorg Med Chem· November 2020

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Combined Peptide and Small-Molecule Approach toward Nonacidic THIQ Inhibitors of the KEAP1/NRF2 Interaction.
Jesus M Ontoria, Ilaria Biancofiore, Paola Fezzardi, Federica Ferrigno, Esther Torrente, Stefania Colarusso

ACS Med Chem Lett· May 2020

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Discovery of (7R)-14-cyclohexyl-7-{[2-(dimethylamino)ethyl](methyl) amino}-7,8-dihydro-6H-indolo[1,2-e][1,5]benzoxazocine-11-carboxylic acid (MK-3281), a potent and orally bioavailable finger-loop inhibitor of the hepatitis C virus NS5B polymerase.
Frank Narjes, Benedetta Crescenzi, Marco Ferrara, Jörg Habermann, Stefania Colarusso

J Med Chem· January 2011

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Optimization of thienopyrrole-based finger-loop inhibitors of the hepatitis C virus NS5B polymerase.
Jose Ignacio Martin Hernando, Jesus Maria Ontoria, Savina Malancona, Barbara Attenni, Fabrizio Fiore, Stefania Colarusso

ChemMedChem· October 2009

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2-(2-Thienyl)-5,6-dihydroxy-4-carboxypyrimidines as inhibitors of the hepatitis C virus NS5B polymerase: discovery, SAR, modeling, and mutagenesis.
Uwe Koch, Barbara Attenni, Savina Malancona, Stefania Colarusso, Immacolata Conte

J Med Chem· March 2006

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Active site inhibitors of HCV NS5B polymerase. The development and pharmacophore of 2-thienyl-5,6-dihydroxypyrimidine-4-carboxylic acid.
Ian Stansfield, Salvatore Avolio, Stefania Colarusso, Nadia Gennari, Frank Narjes

Bioorg Med Chem Lett· October 2004

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SAR and pharmacokinetic studies on phenethylamide inhibitors of the hepatitis C virus NS3/NS4A serine protease.
Savina Malancona, Stefania Colarusso, Jesus M Ontoria, Antonella Marchetti, Marco Poma

Bioorg Med Chem Lett· September 2004

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Phenethyl amides as novel noncovalent inhibitors of hepatitis C virus NS3/4A protease: discovery, initial SAR, and molecular modeling.
Stefania Colarusso, Uwe Koch, Benjamin Gerlach, Christian Steinkühler, Raffaele De Francesco

J Med Chem· January 2003

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A designed P1 cysteine mimetic for covalent and non-covalent inhibitors of HCV NS3 protease.
Frank Narjes, Konrad F Koehler, Uwe Koch, Benjamin Gerlach, Stefania Colarusso

Bioorg Med Chem Lett· February 2002

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Evolution, synthesis and SAR of tripeptide alpha-ketoacid inhibitors of the hepatitis C virus NS3/NS4A serine protease.
Stefania Colarusso, Benjamin Gerlach, Uwe Koch, Ester Muraglia, Immacolata Conte

Bioorg Med Chem Lett· February 2002

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