Publications by authors named "Terry Kenakin"

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Differential Effects of Sodium on Agonist-Induced Conformational Transitions and Signaling at μ and κ Opioid Receptors.
Michael Bram Kuijer, Camryn J Fulton, Talia L Albert, Paloma Knobloch, Jing Wang, Terry Kenakin

Biochemistry· December 2025

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Agonism and Biased Signaling.
Terry Kenakin

Handb Exp Pharmacol· October 2025

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Allosteric modulation of neurotransmission.
Terry Kenakin

Biochem Pharmacol· September 2025

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Differential effects of sodium on agonist-induced conformational transitions and signaling at μ and κ opioid receptors.
Bram Kuijer, Camryn J Fulton, Talia L Albert, Paloma M Knobloch, Jing Wang, Terry Kenakin

bioRxiv· September 2025

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Molecular mechanisms of inverse agonism via κ-opioid receptor-G protein complexes.
Aaliyah S Tyson, Saif Khan, Zenia Motiwala, Gye Won Han, Zixin Zhang, Terry Kenakin

Nat Chem Biol· July 2025

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Know your molecule: pharmacological characterization of drug candidates to enhance efficacy and reduce late-stage attrition.
Terry Kenakin

Nat Rev Drug Discov· August 2024

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Intracellular Allosteric Antagonist of the Olfactory Receptor OR51E2.
Tatjana Abaffy, Olivia Fu, Maira Harume-Nagai, Josh M Goldenberg, Victor Kenyon, Terry Kenakin

Mol Pharmacol· June 2024

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A Pharmacological perspective on the temporal properties of sweeteners.
Guy Servant, Terry Kenakin

Pharmacol Res· June 2024

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Bias translation: The final frontier?
Terry Kenakin

Br J Pharmacol· May 2024

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Allostery: The Good, the Bad, and the Ugly.
Terry Kenakin

J Pharmacol Exp Ther· January 2024

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Neurotensin Receptor Allosterism Revealed in Complex with a Biased Allosteric Modulator.
Brian E Krumm, Jeffrey F DiBerto, Reid H J Olsen, Hye Jin Kang, Samuel T Slocum, Terry Kenakin

Biochemistry· April 2023

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Structural insights into the human niacin receptor HCA2-G signalling complex.
Yang Yang, Hye Jin Kang, Ruogu Gao, Jingjing Wang, Gye Won Han, Terry Kenakin

Nat Commun· March 2023

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Community guidelines for GPCR ligand bias: IUPHAR review 32.
Peter Kolb, Terry Kenakin, Stephen P H Alexander, Marcel Bermudez, Laura M Bohn

Br J Pharmacol· July 2022

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Development of 3-(4-Chlorophenyl)-1-(phenethyl)urea Analogues as Allosteric Modulators of the Cannabinoid Type-1 Receptor: RTICBM-189 is Brain Penetrant and Attenuates Reinstatement of Cocaine-Seeking Behavior.
Thuy Nguyen, Thomas F Gamage, David B Finlay, Ann M Decker, Tiffany L Langston, Terry P Kenakin

J Med Chem· January 2022

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Biased signaling as allosteric probe dependence.
Terry Kenakin

Cell Signal· March 2021

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The function and allosteric control of the human sweet taste receptor.
Guy Servant, Terry Kenakin, Lan Zhang, Mark Williams, Nicole Servant

Adv Pharmacol· September 2020

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Interdependent allosteric free fatty acid receptor 2 modulators synergistically induce functional selective activation and desensitization in neutrophils.
Simon Lind, André Holdfeldt, Jonas Mårtensson, Martina Sundqvist, Terry P Kenakin

Biochim Biophys Acta Mol Cell Res· June 2020

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Virtual discovery of melatonin receptor ligands to modulate circadian rhythms.
Reed M Stein, Hye Jin Kang, John D McCorvy, Grant C Glatfelter, Anthony J Jones, Terry Kenakin

Nature· March 2020

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Emergent Concepts of Receptor Pharmacology.
Terry Kenakin

Handb Exp Pharmacol· January 2020

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G-Protein/Receptor inhibitors as blockers of receptor signaling.
Terry Kenakin

J Theor Biol· November 2019

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Preclinical Testing of Nalfurafine as an Opioid-sparing Adjuvant that Potentiates Analgesia by the Mu Opioid Receptor-targeting Agonist Morphine.
Shane W Kaski, Allison N White, Joshua D Gross, Kristen R Trexler, Kim Wix, Terry Kenakin

J Pharmacol Exp Ther· November 2019

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Discovery and Characterization of a Cellular Potent Positive Allosteric Modulator of the Polycomb Repressive Complex 1 Chromodomain, CBX7.
Kelsey N Lamb, Daniel Bsteh, Sarah N Dishman, Hagar F Moussa, Huitao Fan, Terry P Kenakin

Cell Chem Biol· October 2019

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Can we use Nature's Structure-Activity-Relationships to Make Better Drugs?
Terry Kenakin

Drug Discov Today· September 2019

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Design, Synthesis, and Characterization of Ogerin-Based Positive Allosteric Modulators for G Protein-Coupled Receptor 68 (GPR68).
Xufen Yu, Xi-Ping Huang, Terry P Kenakin, Samuel T Slocum, Xin Chen

J Med Chem· August 2019

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The pharmacologic characterization of allosteric molecules: Gq protein activation.
Sara Bdioui, Julien Verdi, Nicolas Pierre, Eric Trinquet, Thomas Roux, Terry Kenakin

J Recept Signal Transduct Res· April 2019

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