Publications by authors named "Thangeswaran Ramar"

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Prodrug Strategy to Address Impaired Oral Absorption of a Weakly Basic TYK2 Inhibitor Caused by a Gastric Acid-Reducing Agent.
Murugaiah A M Subbaiah, Thangeswaran Ramar, Maheswara Reddy, Sankara Sivaprasad Lvj, Shekhar Yeshwante

J Med Chem· November 2024

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Identification and Optimization of Small Molecule Pyrazolopyrimidine TLR7 Agonists for Applications in Immuno-oncology.
Liqi He, Meng Yao Zhang, Matthew Cox, Qian Zhang, Andrew F Donnell, Thangeswaran Ramar

ACS Med Chem Lett· February 2024

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Promoting Catalytic -Selective Sulfonylation of Cyclopropanols against Conventional -Sulfonylation Using Readily Available Sulfonyl Chlorides.
Thangeswaran Ramar, Andivelu Ilangovan, Murugaiah A M Subbaiah

J Org Chem· October 2023

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Optimization of physicochemical properties of pyrrolidine GPR40 AgoPAMs results in a differentiated profile with improved pharmacokinetics and reduced off-target activities.
Elizabeth A Jurica, Ximao Wu, Kristin N Williams, Lauren E Haque, Richard A Rampulla, Thangeswaran Ramar

Bioorg Med Chem· May 2023

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Electrophilic Hydrazination of Cyclopropanols Using Azodicarboxylates via Copper(II) Catalysis: An Umpolung Strategy to Access β-Hydrazino Ketone Motifs.
Thangeswaran Ramar, Andivelu Ilangovan, Nicholas A Meanwell, Murugaiah A M Subbaiah

J Org Chem· November 2022

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Improving Drug Delivery While Tailoring Prodrug Activation to Modulate and by Optimization of (Carbonyl)oxyalkyl Linker-Based Prodrugs of Atazanavir.
Murugaiah A M Subbaiah, Lakshumanan Subramani, Thangeswaran Ramar, Salil Desai, Sarmistha Sinha

J Med Chem· August 2022

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Orchestrating a β-Hydride Elimination Pathway in Palladium(II)-Catalyzed Arylation/Alkenylation of Cyclopropanols Using Organoboron Reagents.
Thangeswaran Ramar, Murugaiah A M Subbaiah, Andivelu Ilangovan

J Org Chem· April 2022

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(Carbonyl)oxyalkyl linker-based amino acid prodrugs of the HIV-1 protease inhibitor atazanavir that enhance oral bioavailability and plasma trough concentration.
Murugaiah A M Subbaiah, Thangeswaran Ramar, Lakshumanan Subramani, Salil D Desai, Sarmistha Sinha

Eur J Med Chem· December 2020

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Utility of Organoboron Reagents in Arylation of Cyclopropanols via Chelated Pd(II) Catalysis: Chemoselective Access to β-Aryl Ketones.
Thangeswaran Ramar, Murugaiah A M Subbaiah, Andivelu Ilangovan

J Org Chem· June 2020

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Design, Synthesis, and Pharmacokinetic Evaluation of Phosphate and Amino Acid Ester Prodrugs for Improving the Oral Bioavailability of the HIV-1 Protease Inhibitor Atazanavir.
Murugaiah A M Subbaiah, Sandhya Mandlekar, Sridhar Desikan, Thangeswaran Ramar, Lakshumanan Subramani

J Med Chem· April 2019

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Coupling of an Acyl Migration Prodrug Strategy with Bio-activation To Improve Oral Delivery of the HIV-1 Protease Inhibitor Atazanavir.
Murugaiah A M Subbaiah, Nicholas A Meanwell, John F Kadow, Lakshumanan Subramani, Mathiazhagan Annadurai, Thangeswaran Ramar

J Med Chem· May 2018

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Iodine-Mediated C-H Functionalization of sp, sp(2), and sp(3) Carbon: A Unified Multisubstrate Domino Approach for Isatin Synthesis.
Gandhesiri Satish, Ashok Polu, Thangeswaran Ramar, Andivelu Ilangovan

J Org Chem· May 2015

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