Publications by authors named "Timothy D Gross"

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5
5-Aryluracils as potent GnRH antagonists-Characterization of atropisomers.
Liren Zhao, Zhiqiang Guo, Yongsheng Chen, Tao Hu, Dongpei Wu, Timothy D Gross

Bioorg Med Chem Lett· June 2008

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Atropisomeric property of 1-(2,6-difluorobenzyl)-3-[(2R)-amino-2-phenethyl]-5-(2-fluoro-3-methoxyphenyl)-6-methyluracil.
Fabio C Tucci, Tao Hu, Michael F Mesleh, Allan Bokser, Eric Allsopp, Timothy D Gross

Chirality· November 2005

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Uracils as potent antagonists of the human gonadotropin-releasing hormone receptor without atropisomers.
Zhiqiang Guo, Yongsheng Chen, Charles Q Huang, Timothy D Gross, Joseph Pontillo

Bioorg Med Chem Lett· May 2005

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3-[(2R)-Amino-2-phenylethyl]-1-(2,6-difluorobenzyl)-5-(2-fluoro-3-methoxyphenyl)- 6-methylpyrimidin-2,4-dione (NBI 42902) as a potent and orally active antagonist of the human gonadotropin-releasing hormone receptor. Design, synthesis, and in vitro and in vivo characterization.
Fabio C Tucci, Yun-Fei Zhu, R Scott Struthers, Zhiqiang Guo, Timothy D Gross

J Med Chem· February 2005

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Synthesis and structure-activity relationships of uracil derived human GnRH receptor antagonists: (R)-3-[2-(2-amino)phenethyl]-1-(2,6-difluorobenzyl)-6-methyluracils containing a substituted thiophene or thiazole at C-5.
Martin W Rowbottom, Fabio C Tucci, Patrick J Connors, Timothy D Gross, Yun-Fei Zhu

Bioorg Med Chem Lett· October 2004

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3-(2-aminoalkyl)-1-(2,6-difluorobenzyl)-5- (2-fluoro-3-methoxyphenyl)-6-methyl-uracils as orally bioavailable antagonists of the human gonadotropin releasing hormone receptor.
Fabio C Tucci, Yun-Fei Zhu, Zhiqiang Guo, Timothy D Gross, Patrick J Connors

J Med Chem· July 2004

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Synthesis and structure-activity relationships of (R)-1-alkyl-3-[2-(2-amino)phenethyl]-5-(2-fluorophenyl)-6-methyluracils as human GnRH receptor antagonists.
Martin W Rowbottom, Fabio C Tucci, Yun-Fei Zhu, Zhiqiang Guo, Timothy D Gross

Bioorg Med Chem Lett· May 2004

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Synthesis and structure-activity relationships of 1-arylmethyl-5-aryl-6-methyluracils as potent gonadotropin-releasing hormone receptor antagonists.
Zhiqiang Guo, Yun-Fei Zhu, Timothy D Gross, Fabio C Tucci, Yinghong Gao

J Med Chem· February 2004

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Synthesis and structure-activity relationships of 1-arylmethyl-3-(2-aminopropyl)-5-aryl-6-methyluracils as potent GnRH receptor antagonists.
Zhiqiang Guo, Yun-Fei Zhu, Fabio C Tucci, Yinghong Gao, R Scott Struthers, Timothy D Gross

Bioorg Med Chem Lett· October 2003

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Synthesis and structure-activity relationships of 1-arylmethyl-3-(1-methyl-2-amino)ethyl-5-aryl-6-methyluracils as antagonists of the human GnRH Receptor.
Fabio C Tucci, Yun-Fei Zhu, Zhiqiang Guo, Timothy D Gross, Patrick J Connors

Bioorg Med Chem Lett· October 2003

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Identification of 1-arylmethyl-3- (2-aminoethyl)-5-aryluracil as novel gonadotropin-releasing hormone receptor antagonists.
Yun-Fei Zhu, Timothy D Gross, Zhiqiang Guo, Patrick J Connors, Yinghong Gao

J Med Chem· May 2003

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Design and structure-activity relationships of 2-alkyl-3-aminomethyl-6-(3-methoxyphenyl)-7-methyl-8-(2-fluorobenzyl)imidazolo[1,2-a]pyrimid-5-ones as potent GnRH receptor antagonists.
Yun-Fei Zhu, Zhiqiang Guo, Timothy D Gross, Yinghong Gao, Patrick J Connors

J Med Chem· April 2003

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A novel synthesis of 7-aryl-8-fluoro-pyrrolo[1,2-a]pyrimid-4-ones as potent, stable GnRH receptor antagonists.
Fabio C Tucci, Yun-Fei Zhu, Zhiqiang Guo, Timothy D Gross, Patrick J Connors

Bioorg Med Chem Lett· December 2002

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Synthesis and initial structure-activity relationships of a novel series of imidazolo[1,2-a]pyrimid-5-ones as potent GnRH receptor antagonists.
Keith M Wilcoxen, Yun Fei Zhu, Patrick J Connors, John Saunders, Timothy D Gross

Bioorg Med Chem Lett· August 2002

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Design, synthesis and structure-activity relationships of novel imidazolo[1,2-a]pyrimid-5-ones as potent GnRH receptor antagonists.
Timothy D Gross, Yun Fei Zhu, John Saunders, Keith M Wilcoxen, Yinghong Gao

Bioorg Med Chem Lett· August 2002

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Initial structure-activity relationship studies of a novel series of pyrrolo[1,2-a]pyrimid-7-ones as GnRH receptor antagonists.
Yun-Fei Zhu, R Scott Struthers, Patrick J Connors, Yinghong Gao, Timothy D Gross

Bioorg Med Chem Lett· February 2002

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A novel synthesis of 2-arylpyrrolo[1,2-a]pyrimid-7-ones and their structure-activity relationships as potent GnRH receptor antagonists.
Yun-Fei Zhu, Keith Wilcoxen, John Saunders, Zhiqiang Guo, Yinghong Gao, Timothy D Gross

Bioorg Med Chem Lett· February 2002

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