Publications by authors named "Timothy M Chapman"

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Design, synthesis, and biological evaluation of novel pyrrolidinone small-molecule Formyl peptide receptor 2 agonists.
Monika Maciuszek, Almudena Ortega-Gomez, Sanne L Maas, Jose Garrido-Mesa, Bartolo Ferraro, Timothy M Chapman

Eur J Med Chem· December 2021

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Recent advances in the design and development of formyl peptide receptor 2 (FPR2/ALX) agonists as pro-resolving agents with diverse therapeutic potential.
Monika Maciuszek, Antonino Cacace, Eoin Brennan, Catherine Godson, Timothy M Chapman

Eur J Med Chem· March 2021

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Synthesis and evaluation of novel cyclopentane urea FPR2 agonists and their potential application in the treatment of cardiovascular inflammation.
Monika Maciuszek, Almudena Ortega-Gomez, Sanne L Maas, Mauro Perretti, Andy Merritt, Timothy M Chapman

Eur J Med Chem· March 2021

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Design, Synthesis, and Testing of Potent, Selective Hepsin Inhibitors via Application of an Automated Closed-Loop Optimization Platform.
Shishir M Pant, Amanda Mukonoweshuro, Bimbisar Desai, Manoj K Ramjee, Christopher N Selway, Timothy M Chapman

J Med Chem· May 2018

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Imidazopyridazine Inhibitors of Plasmodium falciparum Calcium-Dependent Protein Kinase 1 Also Target Cyclic GMP-Dependent Protein Kinase and Heat Shock Protein 90 To Kill the Parasite at Different Stages of Intracellular Development.
Judith L Green, Robert W Moon, David Whalley, Paul W Bowyer, Claire Wallace, Timothy M Chapman

Antimicrob Agents Chemother· December 2015

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Catechols and 3-hydroxypyridones as inhibitors of the DNA repair complex ERCC1-XPF.
Timothy M Chapman, Kevin J Gillen, Claire Wallace, Maximillian T Lee, Preeti Bakrania

Bioorg Med Chem Lett· October 2015

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N-Hydroxyimides and hydroxypyrimidinones as inhibitors of the DNA repair complex ERCC1-XPF.
Timothy M Chapman, Claire Wallace, Kevin J Gillen, Preeti Bakrania, Puneet Khurana

Bioorg Med Chem Lett· October 2015

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Biochemical and antiparasitic properties of inhibitors of the Plasmodium falciparum calcium-dependent protein kinase PfCDPK1.
Keith H Ansell, Hayley M Jones, David Whalley, Alisdair Hearn, Debra L Taylor, Timothy M Chapman

Antimicrob Agents Chemother· October 2014

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Continuous positive airway pressure (CPAP) during the postoperative period for prevention of postoperative morbidity and mortality following major abdominal surgery.
Claire J Ireland, Timothy M Chapman, Suneeth F Mathew, G Peter Herbison, Mathew Zacharias

Cochrane Database Syst Rev· August 2014

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Optimization of an imidazopyridazine series of inhibitors of Plasmodium falciparum calcium-dependent protein kinase 1 (PfCDPK1).
Timothy M Chapman, Simon A Osborne, Claire Wallace, Kristian Birchall, Nathalie Bouloc

J Med Chem· April 2014

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Substituted imidazopyridazines are potent and selective inhibitors of Plasmodium falciparum calcium-dependent protein kinase 1 (PfCDPK1).
Timothy M Chapman, Simon A Osborne, Nathalie Bouloc, Jonathan M Large, Claire Wallace

Bioorg Med Chem Lett· May 2013

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Substituted aminopyrimidine protein kinase B (PknB) inhibitors show activity against Mycobacterium tuberculosis.
Timothy M Chapman, Nathalie Bouloc, Roger S Buxton, Jasveen Chugh, Kathryn E A Lougheed

Bioorg Med Chem Lett· May 2012

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Ligand-controlled selectivity in the desymmetrization of meso cyclopenten-1,4-diols via rhodium(I)-catalyzed addition of arylboronic acids.
Frederic Menard, David Perez, Daniela Sustac Roman, Timothy M Chapman, Mark Lautens

J Org Chem· June 2010

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Prooxidant activity of oxidized alpha-tocopherol in vegetable oils.
Timothy M Chapman, Hyun Jung Kim, David B Min

J Food Sci· September 2009

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Rhodium-catalyzed asymmetric allylic substitution with boronic acid nucleophiles.
Frederic Menard, Timothy M Chapman, Chris Dockendorff, Mark Lautens

Org Lett· September 2006

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Glyco- and peptidomimetics from three-component Joullié-Ugi coupling show selective antiviral activity.
Timothy M Chapman, Ieuan G Davies, Baohua Gu, Timothy M Block, David I C Scopes

J Am Chem Soc· January 2005

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Highly diastereoselective additions to polyhydroxylated pyrrolidine cyclic imines: ready elaboration of aza-sugar scaffolds to create diverse carbohydrate-processing enzyme probes.
Timothy M Chapman, Steve Courtney, Phil Hay, Benjamin G Davis

Chemistry· July 2003

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Novel cyclic sugar imines: carbohydrate mimics and easily elaborated scaffolds for aza-sugars.
Benjamin G Davis, Michael A T Maughan, Timothy M Chapman, Renaud Villard, Steve Courtney

Org Lett· January 2002

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