Publications by authors named "Variam U Jeankumar"

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Mycobacterium tuberculosis lysine-ɛ-aminotransferase a potential target in dormancy: Benzothiazole based inhibitors.
Rudraraju Srilakshmi Reshma, Variam Ullas Jeankumar, Nidhi Kapoor, Shalini Saxena, Karyakulam Andrews Bobesh

Bioorg Med Chem· May 2017

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Engineering another class of anti-tubercular lead: Hit to lead optimization of an intriguing class of gyrase ATPase inhibitors.
Variam Ullas Jeankumar, Rudraraju Srilakshmi Reshma, Rahul Vats, Renuka Janupally, Shalini Saxena

Eur J Med Chem· October 2016

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Design and development of new class of Mycobacterium tuberculosisl-alanine dehydrogenase inhibitors.
Rudraraju Srilakshmi Reshma, Shalini Saxena, Karyakulam Andrews Bobesh, Variam Ullas Jeankumar, Saritha Gunda

Bioorg Med Chem· September 2016

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Structure-Guided Discovery of Antitubercular Agents That Target the Gyrase ATPase Domain.
Variam U Jeankumar, Shalini Saxena, Rahul Vats, Rudraraju Srilakshmi Reshma, Renuka Janupally

ChemMedChem· March 2016

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Discovery of novel lysine ɛ-aminotransferase inhibitors: An intriguing potential target for latent tuberculosis.
Parthiban Brindha Devi, Jonnalagadda Padma Sridevi, Shruti Singh Kakan, Shalini Saxena, Variam Ullas Jeankumar

Tuberculosis (Edinb)· December 2015

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Design and Biological Evaluation of Furan/Pyrrole/Thiophene-2-carboxamide Derivatives as Efficient DNA GyraseB Inhibitors of Staphylococcus aureus.
Renuka Janupally, Bhramam Medepi, Parthiban Brindha Devi, Priyanka Suryadevara, Variam Ullas Jeankumar

Chem Biol Drug Des· October 2015

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Discovery of potent and selective nonplanar tankyrase inhibiting nicotinamide mimics.
Yves Nkizinkiko, B V S Suneel Kumar, Variam Ullas Jeankumar, Teemu Haikarainen, Jarkko Koivunen

Bioorg Med Chem· August 2015

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Mycobacterial DNA gyrB inhibitors: Ligand based pharmacophore modelling and in vitro enzyme inhibition studies.
Shalini Saxena, Janupally Renuka, Variam Ullas Jeankumar, Perumal Yogeeswari, Dharmarajan Sriram

Curr Top Med Chem· June 2015

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Exploring the gyrase ATPase domain for tailoring newer anti-tubercular drugs: hit to lead optimization of a novel class of thiazole inhibitors.
Variam Ullas Jeankumar, Sonali Kotagiri, Renuka Janupally, Priyanka Suryadevara, Jonnalagadda Padma Sridevi

Bioorg Med Chem· February 2015

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Enabling the (3 + 2) cycloaddition reaction in assembling newer anti-tubercular lead acting through the inhibition of the gyrase ATPase domain: lead optimization and structure activity profiling.
Variam Ullas Jeankumar, Rudraraju Srilakshmi Reshma, Renuka Janupally, Shalini Saxena, Jonnalagadda Padma Sridevi

Org Biomol Chem· February 2015

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A small molecule inhibitor of dengue virus type 2 protease inhibits the replication of all four dengue virus serotypes in cell culture.
Rajendra Raut, Hemalatha Beesetti, Poornima Tyagi, Ira Khanna, Swatantra K Jain, Variam U Jeankumar

Virol J· February 2015

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An efficient synthesis and biological screening of benzofuran and benzo[d]isothiazole derivatives for Mycobacterium tuberculosis DNA GyrB inhibition.
Kummetha Indrasena Reddy, Konduri Srihari, Janupally Renuka, Komanduri Shruthi Sree, Aruna Chuppala, Variam Ullas Jeankumar

Bioorg Med Chem· December 2014

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Development of benzo[d]oxazol-2(3H)-ones derivatives as novel inhibitors of Mycobacterium tuberculosis InhA.
Ganesh S Pedgaonkar, Jonnalagadda Padma Sridevi, Variam Ullas Jeankumar, Shalini Saxena, Parthiban Brindha Devi

Bioorg Med Chem· November 2014

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Structure-guided design and development of novel benzimidazole class of compounds targeting DNA gyraseB enzyme of Staphylococcus aureus.
Renuka Janupally, Variam Ullas Jeankumar, Karyakulam Andrews Bobesh, Vijay Soni, Parthiban Brindha Devi

Bioorg Med Chem· November 2014

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Extending the N-linked aminopiperidine class to the mycobacterial gyrase domain: pharmacophore mapping from known antibacterial leads.
Karyakulam Andrews Bobesh, Janupally Renuka, Variam Ullas Jeankumar, Singh Kakan Shruti, Jonnalagadda Padma Sridevi

Eur J Med Chem· October 2014

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Development of 2-(4-oxoquinazolin-3(4H)-yl)acetamide derivatives as novel enoyl-acyl carrier protein reductase (InhA) inhibitors for the treatment of tuberculosis.
Ganesh S Pedgaonkar, Jonnalagadda Padma Sridevi, Variam Ullas Jeankumar, Shalini Saxena, Parthiban Brindha Devi

Eur J Med Chem· October 2014

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Thiazole-aminopiperidine hybrid analogues: design and synthesis of novel Mycobacterium tuberculosis GyrB inhibitors.
Variam Ullas Jeankumar, Janupally Renuka, Peddi Santosh, Vijay Soni, Jonnalagadda Padma Sridevi

Eur J Med Chem· September 2014

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Design, synthesis, biological evaluation of substituted benzofurans as DNA gyraseB inhibitors of Mycobacterium tuberculosis.
Janupally Renuka, Kummetha Indrasena Reddy, Konduri Srihari, Variam Ullas Jeankumar, Morla Shravan

Bioorg Med Chem· September 2014

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Identification and structure-activity relationship study of carvacrol derivatives as Mycobacterium tuberculosis chorismate mutase inhibitors.
Reshma Alokam, Variam Ullas Jeankumar, Jonnalagadda Padma Sridevi, Siddharth Sai Matikonda, Santosh Peddi

J Enzyme Inhib Med Chem· August 2014

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Gyrase ATPase domain as an antitubercular drug discovery platform: structure-based design and lead optimization of nitrothiazolyl carboxamide analogues.
Variam Ullas Jeankumar, Janupally Renuka, Sonali Kotagiri, Shalini Saxena, Shruti Singh Kakan

ChemMedChem· August 2014

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Discovery and structure optimization of a series of isatin derivatives as Mycobacterium tuberculosis chorismate mutase inhibitors.
Variam U Jeankumar, Reshma Alokam, Jonnalagadda P Sridevi, Priyanka Suryadevara, Siddharth S Matikonda

Chem Biol Drug Des· April 2014

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Development of novel N-linked aminopiperidine-based mycobacterial DNA gyrase B inhibitors: scaffold hopping from known antibacterial leads.
Variam Ullas Jeankumar, Janupally Renuka, Venkat Koushik Pulla, Vijay Soni, Jonnalagadda Padma Sridevi

Int J Antimicrob Agents· March 2014

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Structure-guided design of novel thiazolidine inhibitors of O-acetyl serine sulfhydrylase from Mycobacterium tuberculosis.
Omer Poyraz, Variam Ullas Jeankumar, Shalini Saxena, Robert Schnell, Martin Haraldsson

J Med Chem· August 2013

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Development of 5-nitrothiazole derivatives: identification of leads against both replicative and latent Mycobacterium tuberculosis.
Variam Ullas Jeankumar, Manoj Chandran, Ganesh Samala, Mallika Alvala, Pulla Venkat Koushik

Bioorg Med Chem Lett· December 2012

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Novel acridinedione derivatives: design, synthesis, SIRT1 enzyme and tumor cell growth inhibition studies.
Mallika Alvala, Shubhmita Bhatnagar, Alvala Ravi, Variam Ullas Jeankumar, Thimmappa H Manjashetty

Bioorg Med Chem Lett· May 2012

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