Publications by authors named "Wim Schepens"

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VH antibody loop guides design of a synthetic macrocyclic peptide that potently blocks influenza virus membrane fusion.
Rameshwar U Kadam, Jarek Juraszek, Boerries Brandenburg, Divita Garg, Xueyong Zhu, Wim B G Schepens

Npj Viruses· December 2025

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Discovery of Gut-Restricted PRMT5 Inhibitors to Intercept Colorectal Cancer in Patients with Genetic Loss of Tumor Suppressor Adenomatous Polyposis Coli.
Fabian Hulpia, Wim Schepens, Susan Lepri, Johan Nicolaï, Zhengyu Jiang

J Med Chem· November 2025

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Discovery of Potent and Brain-Penetrant Bicyclic NLRP3 Inhibitors with Peripheral and Central In Vivo Activity.
Oscar Mammoliti, Rodrigo Carbajo, Laura Perez-Benito, Xiaodi Yu, Marion L C Prieri, Wim Schepens

J Med Chem· February 2025

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Discovery and Pharmacological Characterization of JNJ-64619178, a Novel Small-Molecule Inhibitor of PRMT5 with Potent Antitumor Activity.
Dirk Brehmer, Lijs Beke, Tongfei Wu, Hillary J Millar, Christopher Moy, Wim Schepens

Mol Cancer Ther· December 2021

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A small-molecule fusion inhibitor of influenza virus is orally active in mice.
Maria J P van Dongen, Rameshwar U Kadam, Jarek Juraszek, Edward Lawson, Boerries Brandenburg, Wim B G Schepens

Science· March 2019

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Corrigendum to "Chemical space screening around Phe in opioid peptides: Modulating µ versus δ agonism by Suzuki-Miyaura cross-couplings" [Bioorg. Med. Chem. Lett. 28(13) (2018) 2320-2323].
Tom Willemse, Emilie Eiselt, Karlijn Hollanders, Wim Schepens, Herman W T van Vlijmen

Bioorg Med Chem Lett· November 2018

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Chemical space screening around Phe in opioid peptides: Modulating µ versus δ agonism by Suzuki-Miyaura cross-couplings.
Tom Willemse, Emilie Eiselt, Karlijn Hollanders, Wim Schepens, Herman W T van Vlijmen

Bioorg Med Chem Lett· July 2018

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Potent peptidic fusion inhibitors of influenza virus.
Rameshwar U Kadam, Jarek Juraszek, Boerries Brandenburg, Christophe Buyck, Wim B G Schepens

Science· October 2017

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The first one-pot synthesis of L-7-iodotryptophan from 7-iodoindole and serine, and an improved synthesis of other L-7-halotryptophans.
Duncan R M Smith, Tom Willemse, Danai S Gkotsi, Wim Schepens, Bert U W Maes

Org Lett· May 2014

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Design and synthesis of HIV-1 protease inhibitors for a long-acting injectable drug application.
Bart Kesteleyn, Katie Amssoms, Wim Schepens, Geerwin Hache, Wim Verschueren

Bioorg Med Chem Lett· January 2013

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Benzoxazole and benzothiazole amides as novel pharmacokinetic enhancers of HIV protease inhibitors.
Tim H M Jonckers, Marie-Claude Rouan, Geerwin Haché, Wim Schepens, Sabine Hallenberger

Bioorg Med Chem Lett· August 2012

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The development of CD-ring modified analogs of 1alpha,25-dihydroxyvitamin D.
Pierre J De Clercq, Frederik De Buysser, Garrett Minne, Wim Schepens, Freek Vrielynck

J Steroid Biochem Mol Biol· March 2007

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Synthesis of spiro[4.5]decane CF-ring analogues of 1 alpha,25-dihydroxyvitamin D3.
Wim Schepens, Dirk Van Haver, Maurits Vandewalle, Roger Bouillon, Annemieke Verstuyf

Org Lett· September 2006

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Synthesis and biological activity of 22-oxa CD-ring modified analogues of 1alpha,25-dihydroxyvitamin D3: spiro[5.5]undecane CF-ring analogues.
Wim Schepens, Dirk Van Van Haver, Maurits Vandewalle, Pierre J De Clercq, Roger Bouillon

Bioorg Med Chem Lett· August 2004

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