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Publications by authors named "Geerwin Hache"

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Discovery of Potent and Brain-Penetrant Bicyclic NLRP3 Inhibitors with Peripheral and Central In Vivo Activity.
Oscar Mammoliti, Rodrigo Carbajo, Laura Perez-Benito, Xiaodi Yu, Marion L C Prieri, Geerwin Hache

J Med Chem· February 2025


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Spiro-Azetidine Oxindoles as Long-Acting Injectables for Pre-Exposure Prophylaxis against Respiratory Syncytial Virus Infections.
Bart Kesteleyn, Florence Herschke, Nicolas Darville, Bart Stoops, Tom Jacobs, Geerwin Hache

J Med Chem· July 2024


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Design and synthesis of HIV-1 protease inhibitors for a long-acting injectable drug application.
Bart Kesteleyn, Katie Amssoms, Wim Schepens, Geerwin Hache, Wim Verschueren

Bioorg Med Chem Lett· January 2013


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Benzoxazole and benzothiazole amides as novel pharmacokinetic enhancers of HIV protease inhibitors.
Tim H M Jonckers, Marie-Claude Rouan, Geerwin Haché, Wim Schepens, Sabine Hallenberger

Bioorg Med Chem Lett· August 2012


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