Publications by authors named "Angelo Carotti"

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Thioxanthenone-based derivatives as multitarget therapeutic leads for Alzheimer's disease.
Michele Tonelli, Marco Catto, Raimon Sabaté, Valeria Francesconi, Erik Laurini, Angelo Carotti

Eur J Med Chem· March 2023

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Informed Use of 3D-QSAR for the Rational Design of Coumarin Derivatives as Potent and Selective MAO B Inhibitors.
Nicola Gambacorta, Marco Catto, Leonardo Pisani, Angelo Carotti, Orazio Nicolotti

Methods Mol Biol· September 2022

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17β-Hydroxysteroid Dehydrogenase Type 1 Inhibition: A Potential Treatment Option for Non-Small Cell Lung Cancer.
Emanuele M Gargano, Abdelrahman Mohamed, Ahmed S Abdelsamie, Giuseppe F Mangiatordi, Hanna Drzewiecka, Angelo Carotti

ACS Med Chem Lett· December 2021

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Coumarin: A Natural, Privileged and Versatile Scaffold for Bioactive Compounds.
Angela Stefanachi, Francesco Leonetti, Leonardo Pisani, Marco Catto, Angelo Carotti

Molecules· January 2018

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A Round Trip from Medicinal Chemistry to Predictive Toxicology.
Giuseppe Felice Mangiatordi, Angelo Carotti, Ettore Novellino, Orazio Nicolotti

Methods Mol Biol· December 2017

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Potent inhibitors of human LAT1 (SLC7A5) transporter based on dithiazole and dithiazine compounds for development of anticancer drugs.
Lara Napolitano, Mariafrancesca Scalise, Maria Koyioni, Panayiotis Koutentis, Marco Catto, Angelo Carotti

Biochem Pharmacol· November 2017

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Synthesis and Biological Evaluation of Novel Hybrid Molecules Containing Purine, Coumarin and Isoxazoline or Isoxazole Moieties.
Michael G Kallitsakis, Angelo Carotti, Marco Catto, Aikaterini Peperidou, Dimitra J Hadjipavlou-Litina

Open Med Chem J· November 2017

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Indenocinnoline derivatives as G-quadruplex binders, topoisomerase IIα inhibitors and antiproliferative agents.
Grigoris Zoidis, Alice Sosic, Silvia Da Ros, Barbara Gatto, Claudia Sissi, Angelo Carotti

Bioorg Med Chem· May 2017

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3,4-Dihydroquinazoline derivatives inhibit the activities of cholinesterase enzymes.
Byeongyeon Park, Ji Hye Nam, Jin Han Kim, Hyoung Ja Kim, Valentina Onnis, Angelo Carotti

Bioorg Med Chem Lett· March 2017

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Quinolino[3,4-b]quinoxalines and pyridazino[4,3-c]quinoline derivatives: Synthesis, inhibition of topoisomerase IIα, G-quadruplex binding and cytotoxic properties.
Fausta Palluotto, Alice Sosic, Odra Pinato, Grigoris Zoidis, Marco Catto, Angelo Carotti

Eur J Med Chem· November 2016

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Mind the Gap! A Journey towards Computational Toxicology.
Giuseppe Felice Mangiatordi, Domenico Alberga, Cosimo Damiano Altomare, Angelo Carotti, Marco Catto

Mol Inform· September 2016

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Docking-based classification models for exploratory toxicology studies on high-quality estrogenic experimental data.
Daniela Trisciuzzi, Domenico Alberga, Kamel Mansouri, Richard Judson, Saverio Cellamare, Angelo Carotti

Future Med Chem· July 2016

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Exploring Basic Tail Modifications of Coumarin-Based Dual Acetylcholinesterase-Monoamine Oxidase B Inhibitors: Identification of Water-Soluble, Brain-Permeant Neuroprotective Multitarget Agents.
Leonardo Pisani, Roberta Farina, Marco Catto, Rosa Maria Iacobazzi, Orazio Nicolotti, Angelo Carotti

J Med Chem· July 2016

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17β-Hydroxysteroid Dehydrogenase Type 2 Inhibition: Discovery of Selective and Metabolically Stable Compounds Inhibiting Both the Human Enzyme and Its Murine Ortholog.
Emanuele M Gargano, Giuseppe Allegretta, Enrico Perspicace, Angelo Carotti, Chris Van Koppen

PLoS One· April 2016

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Searching for Multi-Targeting Neurotherapeutics against Alzheimer's: Discovery of Potent AChE-MAO B Inhibitors through the Decoration of the 2H-Chromen-2-one Structural Motif.
Leonardo Pisani, Roberta Farina, Ramon Soto-Otero, Nunzio Denora, Giuseppe Felice Mangiatordi, Angelo Carotti

Molecules· March 2016

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Addressing cytotoxicity of 1,4-biphenyl amide derivatives: Discovery of new potent and selective 17β-hydroxysteroid dehydrogenase type 2 inhibitors.
Emanuele Marco Gargano, Enrico Perspicace, Angelo Carotti, Sandrine Marchais-Oberwinkler, Rolf W Hartmann

Bioorg Med Chem Lett· January 2016

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Studies on the antiplatelet and antithrombotic profile of anti-inflammatory coumarin derivatives.
Christos Kontogiorgis, Orazio Nicolotti, Giuseppe Felice Mangiatordi, Massimiliano Tognolini, Foteini Karalaki, Angelo Carotti

J Enzyme Inhib Med Chem· December 2015

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Galloyl benzamide-based compounds modulating tumour necrosis factor α-stimulated c-Jun N-terminal kinase and p38 mitogen-activated protein kinase signalling pathways.
Valentina Leo, Angela Stefanachi, Carmela Nacci, Francesco Leonetti, Modesto de Candia, Angelo Carotti

J Pharm Pharmacol· October 2015

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Structure-Based Design and Optimization of Multitarget-Directed 2H-Chromen-2-one Derivatives as Potent Inhibitors of Monoamine Oxidase B and Cholinesterases.
Roberta Farina, Leonardo Pisani, Marco Catto, Orazio Nicolotti, Domenico Gadaleta, Angelo Carotti

J Med Chem· July 2015

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Multitarget Therapeutic Leads for Alzheimer's Disease: Quinolizidinyl Derivatives of Bi- and Tricyclic Systems as Dual Inhibitors of Cholinesterases and β-Amyloid (Aβ) Aggregation.
Michele Tonelli, Marco Catto, Bruno Tasso, Federica Novelli, Caterina Canu, Angelo Carotti

ChemMedChem· June 2015

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Multitarget-directed tricyclic pyridazinones as G protein-coupled receptor ligands and cholinesterase inhibitors.
Amedeo Pau, Marco Catto, Giovanni Pinna, Simona Frau, Gabriele Murineddu, Angelo Carotti

ChemMedChem· June 2015

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In silico design of novel 2H-chromen-2-one derivatives as potent and selective MAO-B inhibitors.
Leonardo Pisani, Roberta Farina, Orazio Nicolotti, Domenico Gadaleta, Ramon Soto-Otero, Angelo Carotti

Eur J Med Chem· January 2015

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Discovery of new 7-substituted-4-imidazolylmethyl coumarins and 4'-substituted-2-imidazolyl acetophenones open analogues as potent and selective inhibitors of steroid-11β-hydroxylase.
Angela Stefanachi, Nina Hanke, Leonardo Pisani, Francesco Leonetti, Orazio Nicolotti, Angelo Carotti

Eur J Med Chem· January 2015

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Computer-aided structure-based design of multitarget leads for Alzheimer's disease.
José L Domínguez, Fernando Fernández-Nieto, Marian Castro, Marco Catto, M Rita Paleo, Angelo Carotti

J Chem Inf Model· January 2015

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Metabolic stability optimization and metabolite identification of 2,5-thiophene amide 17β-hydroxysteroid dehydrogenase type 2 inhibitors.
Emanuele M Gargano, Enrico Perspicace, Nina Hanke, Angelo Carotti, Sandrine Marchais-Oberwinkler

Eur J Med Chem· November 2014

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