Publications by authors named "Barbara Cosimelli"

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Identification of novel indole derivatives acting as inhibitors of the Keap1-Nrf2 interaction.
Barbara Cosimelli, Giovanni Greco, Sonia Laneri, Ettore Novellino, Antonia Sacchi

J Enzyme Inhib Med Chem· December 2019

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The P-glycoprotein inhibitor diltiazem-like 8-(4-chlorophenyl)-5-methyl-8-[(2Z)-pent-2-en-1-yloxy]-8H-[1,2,4]oxadiazolo[3,4-c][1,4]thiazin-3-one inhibits esterase activity and H3 histone acetylation.
Flavia Cuviello, Faustino Bisaccia, Domenico Spinelli, Maria Francesca Armentano, Sabino Aurelio Bufo, Barbara Cosimelli

Eur J Med Chem· February 2019

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Novel fluorescent triazinobenzimidazole derivatives as probes for labelling human A and A adenosine receptor subtypes.
Elisabetta Barresi, Chiara Giacomelli, Simona Daniele, Ilaria Tonazzini, Marco Robello, Barbara Cosimelli

Bioorg Med Chem· December 2018

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Studies on enantioselectivity of chiral 4-acetylamino-6-alkyloxy-2-alkylthiopyrimidines acting as antagonists of the human A adenosine receptor.
Barbara Cosimelli, Giovanni Greco, Sonia Laneri, Ettore Novellino, Antonia Sacchi

Medchemcomm· January 2018

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4-amino-6-alkyloxy-2-alkylthiopyrimidine derivatives as novel non-nucleoside agonists for the adenosine A receptor.
Barbara Cosimelli, Giovanni Greco, Sonia Laneri, Ettore Novellino, Antonia Sacchi

Chem Biol Drug Des· November 2016

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TSPO-ligands prevent oxidative damage and inflammatory response in C6 glioma cells by neurosteroid synthesis.
Anna Santoro, Giuseppina Mattace Raso, Sabrina Taliani, Eleonora Da Pozzo, Francesca Simorini, Barbara Cosimelli

Eur J Pharm Sci· June 2016

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Enantiomeric 4-Acylamino-6-alkyloxy-2 Alkylthiopyrimidines As Potential A3 Adenosine Receptor Antagonists: HPLC Chiral Resolution and Absolute Configuration Assignment by a Full Set of Chiroptical Spectroscopy.
Daniela Rossi, Rita Nasti, Annamaria Marra, Silvia Meneghini, Giuseppe Mazzeo, Barbara Cosimelli

Chirality· May 2016

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Understanding Oxadiazolothiazinone Biological Properties: Negative Inotropic Activity versus Cytochrome P450-Mediated Metabolism.
Emanuele Carosati, Barbara Cosimelli, Pierfranco Ioan, Elda Severi, Kasiram Katneni

J Med Chem· April 2016

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Deepening the Topology of the Translocator Protein Binding Site by Novel N,N-Dialkyl-2-arylindol-3-ylglyoxylamides.
Elisabetta Barresi, Agostino Bruno, Sabrina Taliani, Sandro Cosconati, Eleonora Da Pozzo, Barbara Cosimelli

J Med Chem· August 2015

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Synthesis and L-type calcium channel blocking activity of new chiral oxadiazolothiazinones.
Emanuele Carosati, Pierfranco Ioan, Giovanni Battista Barrano, Salvatore Caccamese, Barbara Cosimelli

Eur J Med Chem· March 2015

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Osteoblast differentiation and survival: A role for A2B adenosine receptor allosteric modulators.
Maria Letizia Trincavelli, Simona Daniele, Chiara Giacomelli, Sabrina Taliani, Federico Da Settimo, Barbara Cosimelli

Biochim Biophys Acta· December 2014

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Playing with opening and closing of heterocycles: using the cusmano-ruccia reaction to develop a novel class of oxadiazolothiazinones, active as calcium channel modulators and P-glycoprotein inhibitors.
Domenico Spinelli, Roberta Budriesi, Barbara Cosimelli, Elda Severi, Matteo Micucci

Molecules· October 2014

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Synthesis and biological evaluation of imidazo[1,2-a]pyrimidines and imidazo[1,2-a]pyridines as new inhibitors of the Wnt/β-catenin signaling.
Barbara Cosimelli, Sonia Laneri, Carmine Ostacolo, Antonia Sacchi, Elda Severi

Eur J Med Chem· August 2014

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p53 functional inhibitors behaving like pifithrin-β counteract the Alzheimer peptide non-β-amyloid component effects in human SH-SY5Y cells.
Eleonora Da Pozzo, Valeria La Pietra, Barbara Cosimelli, Federico Da Settimo, Chiara Giacomelli

ACS Chem Neurosci· May 2014

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Allosteric modulators of human A2B adenosine receptor.
Maria Letizia Trincavelli, Chiara Giacomelli, Simona Daniele, Sabrina Taliani, Barbara Cosimelli

Biochim Biophys Acta· March 2014

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Modulation of A2B adenosine receptor by 1-Benzyl-3-ketoindole derivatives.
Sabrina Taliani, Maria Letizia Trincavelli, Barbara Cosimelli, Sonia Laneri, Elda Severi

Eur J Med Chem· November 2013

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ABCB1 Structural Models, Molecular Docking, and Synthesis of New Oxadiazolothiazin-3-one Inhibitors.
Camillo Rosano, Maurizio Viale, Barbara Cosimelli, Elda Severi, Rosaria Gangemi

ACS Med Chem Lett· August 2013

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Absolute configuration and biological profile of two thiazinooxadiazol-3-ones with L-type calcium channel activity: a study of the structural effects.
Pierfranco Ioan, Alessia Ciogli, Francesco Sirci, Roberta Budriesi, Barbara Cosimelli

Org Biomol Chem· December 2012

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From the pharmacophore to the homology model of the benzodiazepine receptor: the indolyglyoxylamides affair.
Barbara Cosimelli, Sandro Cosconati, Luciana Marinelli, Ettore Novellino, Giovanni Greco

Curr Top Med Chem· June 2012

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3-aryl-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-one: a novel template for the design of highly selective A₂B adenosine receptor antagonists.
Sabrina Taliani, Isabella Pugliesi, Elisabetta Barresi, Francesca Simorini, Silvia Salerno, Barbara Cosimelli

J Med Chem· February 2012

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Derivatives of benzimidazol-2-ylquinoline and benzimidazol-2-ylisoquinoline as selective A1 adenosine receptor antagonists with stimulant activity on human colon motility.
Barbara Cosimelli, Sabrina Taliani, Giovanni Greco, Ettore Novellino, Annalisa Sala

ChemMedChem· October 2011

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Tertiary amides with a five-membered heteroaromatic ring as new probes for the translocator protein.
Barbara Cosimelli, Francesca Simorini, Sabrina Taliani, Concettina La Motta, Federico Da Settimo

Eur J Med Chem· September 2011

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Preliminary finding on a new calcium channel entry blocker chemotype: 5,6-diamino-4-hydroxy-2-mercaptopyrimidine derivatives.
Barbara Cosimelli, Elda Severi, Ettore Novellino, Anna Cavaccini, Mauro Cataldi

J Med Chem· August 2011

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Novel N2-substituted pyrazolo[3,4-d]pyrimidine adenosine A3 receptor antagonists: inhibition of A3-mediated human glioblastoma cell proliferation.
Sabrina Taliani, Concettina La Motta, Laura Mugnaini, Francesca Simorini, Silvia Salerno, Barbara Cosimelli

J Med Chem· May 2010

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Novel irreversible fluorescent probes targeting the 18 kDa translocator protein: synthesis and biological characterization.
Sabrina Taliani, Eleonora Da Pozzo, Marusca Bellandi, Sara Bendinelli, Isabella Pugliesi, Barbara Cosimelli

J Med Chem· May 2010

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