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Publications by authors named "Benjamin Doerfel"

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Phenotypic Hit Identification and Optimization of Novel Pan-TEAD and Subtype-Selective Inhibitors.
Timo Heinrich, Alessia Gambardella, Daniel Schwarz, Carl Petersson, Jakub Gunera, Benjamin Doerfel

J Med Chem· November 2025


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MoA Studies of the TEAD P-Site Binding Ligand MSC-4106 and Its Optimization to TEAD1-Selective Amide M3686.
Timo Heinrich, Daniel Schwarz, Carl Petersson, Jakub Gunera, Sakshi Garg, Benjamin Doerfel

J Med Chem· March 2025


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Selective Wee1 Inhibitors Led to Antitumor Activity and Correlated with Myelosuppression.
Satenig Guler, Maria C DiPoto, Alejandro Crespo, Richard Caldwell, Benjamin Doerfel

ACS Med Chem Lett· May 2023


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Optimization of TEAD P-Site Binding Fragment Hit into In Vivo Active Lead .
Timo Heinrich, Carl Peterson, Richard Schneider, Sakshi Garg, Daniel Schwarz, Benjamin Doerfel

J Med Chem· July 2022


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