Publications by authors named "Colin R Rose"

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Discovery of SARS-CoV-2 papain-like protease (PL) inhibitors with efficacy in a murine infection model.
Michelle R Garnsey, Matthew C Robinson, Luong T Nguyen, Rhonda Cardin, Joseph Tillotson, Colin R Rose

Sci Adv· August 2024

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6-Azaspiro[2.5]octanes as small molecule agonists of the human glucagon-like peptide-1 receptor.
Gary E Aspnes, Scott W Bagley, Steven B Coffey, Edward L Conn, John M Curto, Colin R Rose

Bioorg Med Chem Lett· October 2023

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Preparation of Azinones from (Cyclopropylmethoxy)azine Ethers.
Allyn T Londregan, John M Curto, Emma Hastry, Colin R Rose, Simon Berritt

J Org Chem· May 2023

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A General Synthesis of Dihydronaphthyridinones with Aryl-Substituted Quaternary Benzylic Centers.
John C Murray, Colin R Rose, John M Curto

J Org Chem· March 2023

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Highly potent and selective Na1.7 inhibitors for use as intravenous agents and chemical probes.
R Ian Storer, Andy Pike, Nigel A Swain, Aristos J Alexandrou, Bruce M Bechle, Colin R Rose

Bioorg Med Chem Lett· November 2017

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One-Pot Synthesis of α-Branched N-Acylamines via Titanium-Mediated Condensation of Amides, Aldehydes, and Organometallics.
Chunhui Dai, Julien Genovino, Bruce M Bechle, Matthew S Corbett, Chan Woo Huh, Colin R Rose

Org Lett· March 2017

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Practical synthesis of capromorelin, a growth hormone secretagogue, via a crystallization-induced dynamic resolution.
Colin R Rose, Michael P Zawistoski, Bruce A Lefker, F Michael Mangano, Ann S Wright

Bioorg Med Chem· February 2017

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Discovery and Preclinical Characterization of 6-Chloro-5-[4-(1-hydroxycyclobutyl)phenyl]-1H-indole-3-carboxylic Acid (PF-06409577), a Direct Activator of Adenosine Monophosphate-activated Protein Kinase (AMPK), for the Potential Treatment of Diabetic Nephropathy.
Kimberly O Cameron, Daniel W Kung, Amit S Kalgutkar, Ravi G Kurumbail, Russell Miller, Colin R Rose

J Med Chem· September 2016

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Design and development of histone deacetylase (HDAC) chemical probes for cell-based profiling.
Victoria E Albrow, Rachel L Grimley, James Clulow, Colin R Rose, Jianmin Sun

Mol Biosyst· May 2016

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The Synthesis of Methyl-Substituted Spirocyclic Piperidine-Azetidine (2,7-Diazaspiro[3.5]nonane) and Spirocyclic Piperidine-Pyrrolidine (2,8-Diazaspiro[4.5]decane) Ring Systems.
Aaron C Smith, Shawn Cabral, Daniel W Kung, Colin R Rose, James A Southers

J Org Chem· May 2016

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Diastereoselective synthesis of β-heteroaryl syn-α-methyl-β-amino acid derivatives via a double chiral auxiliary approach.
Jianwei Bian, David Blakemore, Joseph S Warmus, Jianmin Sun, Matthew Corbett, Colin R Rose

Org Lett· February 2013

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Identification of spirocyclic piperidine-azetidine inverse agonists of the ghrelin receptor.
Daniel W Kung, Steven B Coffey, Ryan M Jones, Shawn Cabral, Wenhua Jiao, Colin R Rose

Bioorg Med Chem Lett· July 2012

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Synthesis of 7-oxo-dihydrospiro[indazole-5,4'-piperidine] acetyl-CoA carboxylase inhibitors.
Scott W Bagley, James A Southers, Shawn Cabral, Colin R Rose, David J Bernhardson

J Org Chem· February 2012

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Discovery and evaluation of pyrazolo[1,5-a]pyrimidines as neuropeptide Y1 receptor antagonists.
David A Griffith, Diane M Hargrove, Tristan S Maurer, Charles A Blum, Stéphane De Lombaert, Colin R Rose

Bioorg Med Chem Lett· May 2011

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New bicyclic cannabinoid receptor-1 (CB1-R) antagonists.
Philip A Carpino, David A Griffith, Subas Sakya, Robert L Dow, Shawn C Black, Colin R Rose

Bioorg Med Chem Lett· February 2006

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Pyrazolinone-piperidine dipeptide growth hormone secretagogues (GHSs). Discovery of capromorelin.
Philip A Carpino, Bruce A Lefker, Steven M Toler, Lydia C Pan, John R Hadcock, Colin R Rose

Bioorg Med Chem· February 2003

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Discovery and biological characterization of capromorelin analogues with extended half-lives.
Philip A Carpino, Bruce A Lefker, Steven M Toler, Lydia C Pan, John R Hadcock, Colin R Rose

Bioorg Med Chem Lett· November 2002

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