Publications by authors named "Derek Cogan"

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Pharmacodynamic effects of highly selective aldosterone synthase inhibitor vicadrostat in cynomolgus monkeys: Contrasting effects of once versus twice daily dosing.
Steven M Weldon, Derek A Cogan, Matthew A Cerny, Kosea S Frederick, Kristina K Gueneva-Boucheva

J Pharmacol Exp Ther· August 2025

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Targeting chromosomally unstable tumors with a selective KIF18A inhibitor.
Aaron F Phillips, Rumin Zhang, Mia Jaffe, Ryan Schulz, Marysol Chu Carty, Derek A Cogan

Nat Commun· January 2025

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Re-awakening Innate Immune Signaling in Cancer: The Development of Highly Potent ENPP1 Inhibitors.
Derek Cogan, Samuel F Bakhoum

Cell Chem Biol· November 2020

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Dihydrobenzisoxazole-4-one compounds are novel selective inhibitors of aldosterone synthase (CYP11B2) with in vivo activity.
Kenneth Meyers, Derek A Cogan, Jennifer Burke, Raquel Arenas, Michael Balestra

Bioorg Med Chem Lett· March 2018

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N-Arylsulfonyl-α-amino carboxamides are potent and selective inhibitors of the chemokine receptor CCR10 that show efficacy in the murine DNFB model of contact hypersensitivity.
Asitha Abeywardane, Gary Caviness, Younggi Choi, Derek Cogan, Amy Gao

Bioorg Med Chem Lett· November 2016

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Selectivity of BI 689648, a Novel, Highly Selective Aldosterone Synthase Inhibitor: Comparison with FAD286 and LCI699 in Nonhuman Primates.
Steven M Weldon, Matthew A Cerny, Kristina Gueneva-Boucheva, Derek Cogan, Xin Guo

J Pharmacol Exp Ther· October 2016

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Exploration of cathepsin S inhibitors characterized by a triazole P1-P2 amide replacement.
Neil Moss, Zhaoming Xiong, Mike Burke, Derek Cogan, Donghong A Gao

Bioorg Med Chem Lett· December 2012

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Indole RSK inhibitors. Part 1: discovery and initial SAR.
Stephen J Boyer, Jennifer Burke, Xin Guo, Thomas M Kirrane, Roger J Snow, Derek Cogan

Bioorg Med Chem Lett· January 2012

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A new class of 5-HT2B antagonists possesses favorable potency, selectivity, and rat pharmacokinetic properties.
Neil Moss, Younggi Choi, Derek Cogan, Adam Flegg, Andreas Kahrs

Bioorg Med Chem Lett· April 2009

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Synthesis and SAR studies of indole-based MK2 inhibitors.
Zhaoming Xiong, Donghong Amy Gao, Derek A Cogan, Daniel R Goldberg, Ming-Hong Hao

Bioorg Med Chem Lett· March 2008

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Discovery of potent and selective PKC-theta inhibitors.
Charles L Cywin, Georg Dahmann, Anthony S Prokopowicz, Erick R R Young, Ronald L Magolda, Derek A Cogan

Bioorg Med Chem Lett· January 2007

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