Publications by authors named "Dina Manetti"

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Ibogalogs decrease neuropathic pain in mice through a mechanism involving crosstalk between 5-HT and mGlu receptors.
Hugo R Arias, Laura Micheli, Anders A Jensen, Sonya Galant, Franck Vandermoere, Dina Manetti

Biomed Pharmacother· March 2025

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The psychoplastogens ibogaminalog and ibogainalog induce antidepressant-like activity in naïve and depressed mice by mechanisms involving 5-HT receptor activation and serotonergic transmission.
Hugo R Arias, Deborah Rudin, Dino Luethi, Jan Valenta, Anna Leśniak, Dina Manetti

Prog Neuropsychopharmacol Biol Psychiatry· January 2025

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Novel psychoplastogen DM506 reduces cue-induced heroin-seeking and inhibits tonic GABA currents in the Prelimbic Cortex.
Kassandra Looschen, Shailesh Narayan Khatri, Malabika Maulik, Colin Salisbury, Alaina F Carman, Dina Manetti

Neurochem Int· September 2024

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Non-hallucinogenic compounds derived from iboga alkaloids alleviate neuropathic and visceral pain in mice through a mechanism involving 5-HT receptor activation.
Hugo R Arias, Laura Micheli, Deborah Rudin, Ophelie Bento, Saskia Borsdorf, Dina Manetti

Biomed Pharmacother· August 2024

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Dual Inhibitors of P-gp and Carbonic Anhydrase XII (hCA XII) against Tumor Multidrug Resistance with Piperazine Scaffold.
Laura Braconi, Chiara Riganti, Astrid Parenti, Marta Cecchi, Alessio Nocentini, Dina Manetti

Molecules· July 2024

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The novel non-hallucinogenic compound DM506 (3-methyl-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole) induces sedative- and anxiolytic-like activity in mice by a mechanism involving 5-HT receptor activation.
Hugo R Arias, Deborah Rudin, Dustin J Hines, April Contreras, Alican Gulsevin, Dina Manetti

Eur J Pharmacol· March 2024

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Synthetic Approaches to Piperazine-Containing Drugs Approved by FDA in the Period of 2011-2023.
Maria Novella Romanelli, Laura Braconi, Alessio Gabellini, Dina Manetti, Giambattista Marotta

Molecules· December 2023

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Tetrazole and oxadiazole derivatives as bioisosteres of tariquidar and elacridar: New potent P-gp modulators acting as MDR reversers.
Laura Braconi, Silvia Dei, Marialessandra Contino, Chiara Riganti, Gianluca Bartolucci, Dina Manetti

Eur J Med Chem· November 2023

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The Antinociceptive Activity of (E)-3-(thiophen-2-yl)- N -(p-tolyl)acrylamide in Mice Is Reduced by (E)-3-(furan-2-yl)- N -methyl- N -(p-tolyl)acrylamide Through Opposing Modulatory Mechanisms at the α7 Nicotinic Acetylcholine Receptor.
Hugo R Arias, Han-Shen Tae, Laura Micheli, Arsalan Yousuf, Dina Manetti

Anesth Analg· September 2023

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Chemical, Pharmacological, and Structural Characterization of Novel Acrylamide-Derived Modulators of the GABA Receptor.
Hugo R Arias, Spencer R Pierce, Allison L Germann, Sophia Q Xu, Marcelo O Ortells, Dina Manetti

Mol Pharmacol· September 2023

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DM506 (3-Methyl-1,2,3,4,5,6-hexahydroazepino[4,5-]indole fumarate), a Novel Derivative of Ibogamine, Inhibits α7 and α9α10 Nicotinic Acetylcholine Receptors by Different Allosteric Mechanisms.
Han-Shen Tae, Marcelo O Ortells, Bassel J Tekarli, Dina Manetti, Maria Novella Romanelli

ACS Chem Neurosci· July 2023

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The Tetrahydroisoquinoline Scaffold in ABC Transporter Inhibitors that Act as Multidrug Resistance (MDR) Reversers.
Elisabetta Teodori, Laura Braconi, Dina Manetti, Maria Novella Romanelli, Silvia Dei

Curr Top Med Chem· January 2023

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Recent Advances in the Discovery of Nicotinic Acetylcholine Receptor Allosteric Modulators.
Dina Manetti, Silvia Dei, Hugo R Arias, Laura Braconi, Alessio Gabellini

Molecules· January 2023

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New Dual P-Glycoprotein (P-gp) and Human Carbonic Anhydrase XII (hCA XII) Inhibitors as Multidrug Resistance (MDR) Reversers in Cancer Cells.
Laura Braconi, Elisabetta Teodori, Chiara Riganti, Marcella Coronnello, Alessio Nocentini, Dina Manetti

J Med Chem· November 2022

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The piperazine scaffold for novel drug discovery efforts: the evidence to date.
Maria Novella Romanelli, Dina Manetti, Laura Braconi, Silvia Dei, Alessio Gabellini

Expert Opin Drug Discov· September 2022

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Overcoming Multidrug Resistance (MDR): Design, Biological Evaluation and Molecular Modelling Studies of 2,4-Substituted Quinazoline Derivatives.
Laura Braconi, Elisabetta Teodori, Marialessandra Contino, Chiara Riganti, Gianluca Bartolucci, Dina Manetti

ChemMedChem· June 2022

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Type I and type II positive allosteric modulators of α7 nicotinic acetylcholine receptors induce antidepressant-like activity in mice by a mechanism involving receptor potentiation but not neurotransmitter reuptake inhibition. Correlation with mTOR intracellular pathway activation.
Katarzyna M Targowska-Duda, Barbara Budzynska, Agnieszka Michalak, Artur Wnorowski, Claus J Loland, Dina Manetti

Eur Neuropsychopharmacol· November 2021

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6,7-Dimethoxy-2-phenethyl-1,2,3,4-tetrahydroisoquinoline amides and corresponding ester isosteres as multidrug resistance reversers.
Laura Braconi, Gianluca Bartolucci, Marialessandra Contino, Niccolò Chiaramonte, Roberta Giampietro, Dina Manetti

J Enzyme Inhib Med Chem· December 2020

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()-3-Furan-2-yl---tolyl-acrylamide and its Derivative DM489 Decrease Neuropathic Pain in Mice Predominantly by α7 Nicotinic Acetylcholine Receptor Potentiation.
Hugo R Arias, Carla Ghelardini, Elena Lucarini, Han-Shen Tae, Arsalan Yousuf, Dina Manetti

ACS Chem Neurosci· November 2020

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Carbachol dimers with primary carbamate groups as homobivalent modulators of muscarinic receptors.
Rosanna Matucci, Cristina Bellucci, Maria Vittoria Martino, Marta Nesi, Dina Manetti

Eur J Pharmacol· September 2020

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Dual P-Glycoprotein and CA XII Inhibitors: A New Strategy to Reverse the P-gp Mediated Multidrug Resistance (MDR) in Cancer Cells.
Elisabetta Teodori, Laura Braconi, Silvia Bua, Andrea Lapucci, Gianluca Bartolucci, Dina Manetti

Molecules· April 2020

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Design, synthesis and biological evaluation of stereo- and regioisomers of amino aryl esters as multidrug resistance (MDR) reversers.
Elisabetta Teodori, Marialessandra Contino, Chiara Riganti, Gianluca Bartolucci, Laura Braconi, Dina Manetti

Eur J Med Chem· November 2019

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Modulation of the spacer in N,N-bis(alkanol)amine aryl ester heterodimers led to the discovery of a series of highly potent P-glycoprotein-based multidrug resistance (MDR) modulators.
Silvia Dei, Laura Braconi, Alfonso Trezza, Marta Menicatti, Marialessandra Contino, Dina Manetti

Eur J Med Chem· June 2019

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EC18 as a Tool To Understand the Role of HCN4 Channels in Mediating Hyperpolarization-Activated Current in Tissues.
Maria Novella Romanelli, Martina Del Lungo, Luca Guandalini, Mehrnoush Zobeiri, András Gyökeres, Dina Manetti

ACS Med Chem Lett· April 2019

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New Rigid Nicotine Analogues, Carrying a Norbornane Moiety, Are Potent Agonists of α7 and α3* Nicotinic Receptors.
Dina Manetti, Alexandra Garifulina, Gianluca Bartolucci, Carla Bazzicalupi, Cristina Bellucci

J Med Chem· February 2019

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