Publications by authors named "Dominique Perrin"

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Comparative analysis of YAP/TEAD inhibitors in 2D and 3D cultures of primary human hepatocytes reveals a novel non-canonical mechanism of CYP induction.
Nuria Oliva-Vilarnau, Sabine U Vorrink, Florian A Büttner, Timo Heinrich, Janike Sensbach, Dominique Perrin

Biochem Pharmacol· September 2023

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Assessment of the potential of the MET inhibitor tepotinib to affect the pharmacokinetics of CYP3A4 and P-gp substrates.
Özkan Yalkinoglu, Andreas Becker, Axel Krebs-Brown, Claudia Vetter, Christian Lüpfert, Dominique Perrin

Invest New Drugs· August 2023

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IOA-244 is a Non-ATP-competitive, Highly Selective, Tolerable PI3K Delta Inhibitor That Targets Solid Tumors and Breaks Immune Tolerance.
Zoë Johnson, Chiara Tarantelli, Elisa Civanelli, Luciano Cascione, Filippo Spriano, Dominique Perrin

Cancer Res Commun· April 2023

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Differences in Sustained Cellular Effects of MET inhibitors Are Driven by Prolonged Target Engagement and Lysosomal Retention.
Nina Berges, Jan Henrik Klug, Anna Eicher, Jennifer Loehr, Daniel Schwarz, Dominique Perrin

Mol Pharmacol· February 2023

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Brain penetration and efficacy of tepotinib in orthotopic patient-derived xenograft models of MET-driven non-small cell lung cancer brain metastases.
Manja Friese-Hamim, Anderson Clark, Dominique Perrin, Lindsey Crowley, Christof Reusch

Lung Cancer· January 2022

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Insights into Praziquantel Metabolism and Potential Enantiomeric Cytochrome P450-Mediated Drug-Drug Interaction.
Gloria Vendrell-Navarro, Holger Scheible, Floriane Lignet, Howard Burt, Christian Luepfert, Dominique Perrin

Drug Metab Dispos· June 2020

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Comparison of methods for the prediction of human clearance from hepatocyte intrinsic clearance for a set of reference compounds and an external evaluation set.
Tetsuo Yamagata, Ugo Zanelli, Dieter Gallemann, Dominique Perrin, Hugues Dolgos

Xenobiotica· September 2017

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Hepatoprotective and antidiabetic effects of Pistacia lentiscus leaf and fruit extracts.
Chafiaâ Mehenni, Dina Atmani-Kilani, Stéphane Dumarçay, Dominique Perrin, Philippe Gérardin

J Food Drug Anal· July 2016

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Capillary microfluidic electrophoretic mobility shift assays: application to enzymatic assays in drug discovery.
Dominique Perrin, Christèle Frémaux, Adam Shutes

Expert Opin Drug Discov· January 2010

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Pelvic abscess associated with Haemophilus influenzae bacteremia.
Gilles Guerrier, Laurent Morisse, Dominique Perrin

Int J Gynaecol Obstet· November 2009

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GLEPP1/protein-tyrosine phosphatase phi inhibitors block chemotaxis in vitro and in vivo and improve murine ulcerative colitis.
Rosanna Pescini Gobert, Monique van den Eijnden, Cedric Szyndralewiez, Catherine Jorand-Lebrun, Dominique Swinnen, Dominique Perrin

J Biol Chem· April 2009

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Convergent functional genomics of oligodendrocyte differentiation identifies multiple autoinhibitory signaling circuits.
Rosanna Pescini Gobert, Lara Joubert, Marie-Laure Curchod, Catherine Salvat, Isabelle Foucault, Dominique Perrin

Mol Cell Biol· March 2009

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In vitro and in vivo pharmacological profile of AS057278, a selective d-amino acid oxidase inhibitor with potential anti-psychotic properties.
Tiziana Adage, Anne-Cécile Trillat, Anna Quattropani, Dominique Perrin, Laurent Cavarec

Eur Neuropsychopharmacol· March 2008

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Protein-tyrosine phosphatase H1 controls growth hormone receptor signaling and systemic growth.
Iwona Pilecka, Claudia Patrignani, Rosanna Pescini, Marie-Laure Curchod, Dominique Perrin

J Biol Chem· November 2007

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Structural basis for selective inhibition of Mycobacterium tuberculosis protein tyrosine phosphatase PtpB.
Christoph Grundner, Dominique Perrin, Rob Hooft van Huijsduijnen, Dominique Swinnen, Jérome Gonzalez

Structure· April 2007

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A microfluidics-based mobility shift assay to discover new tyrosine phosphatase inhibitors.
Dominique Perrin, Christèle Frémaux, Dominique Besson, Wolfgang H B Sauer, Alexander Scheer

J Biomol Screen· December 2006

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Assay development and screening of a serine/threonine kinase in an on-chip mode using caliper nanofluidics technology.
Dominique Perrin, Christèle Frémaux, Alexander Scheer

J Biomol Screen· June 2006

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Furan-2-ylmethylene thiazolidinediones as novel, potent, and selective inhibitors of phosphoinositide 3-kinase gamma.
Vincent Pomel, Jasna Klicic, David Covini, Dennis D Church, Jeffrey P Shaw, Dominique Perrin

J Med Chem· June 2006

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Overcoming the hurdle of fluorescent compounds in kinase screening: a case study.
Dominique Perrin, Thierry Martin, Yves Cambet, Christèle Frémaux, Alexander Scheer

Assay Drug Dev Technol· April 2006

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Soil organic carbon changes in landscape units of Belgium between 1960 and 2000 with reference to 1990.
Suzanna Lettens, Jos VAN Orshoven, Bas VAN Wesemael, Bart Muys, Dominique Perrin

Glob Chang Biol· December 2005

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Blockade of PI3Kgamma suppresses joint inflammation and damage in mouse models of rheumatoid arthritis.
Montserrat Camps, Thomas Rückle, Hong Ji, Vittoria Ardissone, Felix Rintelen, Dominique Perrin

Nat Med· September 2005

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Comparison of 8 vs 15 days of antibiotic therapy for ventilator-associated pneumonia in adults: a randomized trial.
Jean Chastre, Michel Wolff, Jean-Yves Fagon, Sylvie Chevret, Franck Thomas, Dominique Perrin

JAMA· November 2003

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A homogeneous 384-well high-throughput binding assay for a TNF receptor using alphascreen technology.
Janet Wilson, Claudia Pena Rossi, Susanna Carboni, Christèle Fremaux, Dominique Perrin

J Biomol Screen· October 2003

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Apoptotic cell death induction by F 11782 a novel dual catalytic inhibitor of topoisomerases I and II.
Chantal Etiévant, Anna Kruczynski, Jean-Marc Barret, Dominique Perrin, Bridget T Hill

Biochem Pharmacol· March 2003

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Increased endogenous carbon monoxide production in severe sepsis.
Rachid Zegdi, Dominique Perrin, Michèle Burdin, Richard Boiteau, Alain Tenaillon

Intensive Care Med· June 2002

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