Publications by authors named "Frederic Rodriguez"

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Is Mycobacterial InhA a Suitable Target for Rational Drug Design?
Julien Rizet, Laurent Maveyraud, David Rengel, Valérie Guillet, Gabriel Publicola, Frédéric Rodriguez

ChemMedChem· July 2025

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Repression of Connexin26 hemichannel activity protects the barrier function of respiratory airway epithelial cells against LPS-induced alteration.
Tina Lehrich, Anne Dierks, Masina Plenge, Helena Obernolte, Klaudia Grieger, Frederic Rodriguez

Cell Commun Signal· May 2025

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Imidazoquinoline Derivatives as Potential Inhibitors of InhA Enzyme and .
Pascal Hoffmann, Joëlle Azéma-Despeyroux, Fernanda Goncalves, Alessandro Stamilla, Nathalie Saffon-Merceron, Frédéric Rodriguez

Molecules· June 2024

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Multivalent pyrrolidines acting as pharmacological chaperones against Gaucher disease.
Marc Borie-Guichot, My Lan Tran, Virginie Garcia, Abdelouahd Oukhrib, Frédéric Rodriguez

Bioorg Chem· May 2024

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Exploring the plasticity of the InhA substrate-binding site using new diaryl ether inhibitors.
Rasoul Tamhaev, Emeline Grosjean, Hikmat Ahamed, Mélina Chebaiki, Frédéric Rodriguez

Bioorg Chem· February 2024

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Discovery of new diaryl ether inhibitors against Mycobacterium tuberculosis targeting the minor portal of InhA.
Mélina Chebaiki, Evelyne Delfourne, Rasoul Tamhaev, Saïda Danoun, Frédéric Rodriguez

Eur J Med Chem· November 2023

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Phenyl dialkynylcarbinols, a Bioinspired Series of Synthetic Antitumor Acetylenic Lipids.
Margaux Bossuat, Pauline Rullière, Nadège Preuilh, Antonio Peixoto, Etienne Joly, Frédéric Rodriguez

J Med Chem· October 2023

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IDO1 and TDO inhibitory evaluation of analogues of the marine pyrroloiminoquinone alkaloids: Wakayin and Tsitsikammamines.
Thomas Levy, Laura Marchand, Vincent Stroobant, Luc Pilotte, Benoît Van den Eynde, Frédéric Rodriguez

Bioorg Med Chem Lett· May 2021

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Isolation and identification of ten new sildenafil derivatives in an alleged herbal supplement for sexual enhancement.
Gaëtan Assemat, Stéphane Balayssac, Véronique Gilard, Nathalie Martins-Froment, Isabelle Fabing, Frédéric Rodriguez

J Pharm Biomed Anal· November 2020

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Concise asymmetric synthesis of new enantiomeric -alkyl pyrrolidines acting as pharmacological chaperones against Gaucher disease.
Tessa Castellan, Virginie Garcia, Frédéric Rodriguez, Isabelle Fabing, Yevhenii Shchukin

Org Biomol Chem· October 2020

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N,O-Dialkyl deoxynojirimycin derivatives as CERT START domain ligands.
Tessa Castellan, Cécile Santos, Frédéric Rodriguez, Mathieu L Lepage, Yan Liang

Bioorg Med Chem Lett· January 2020

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First triclosan-based macrocyclic inhibitors of InhA enzyme.
Frédéric Rodriguez, Nathalie Saffon, José Camilla Sammartino, Giulia Degiacomi, Maria Rosalia Pasca

Bioorg Chem· January 2020

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Modification of endothelial nitric oxide synthase by 4-oxo-2(E)-nonenal(ONE) in preeclamptic placentas.
Paul Guerby, Audrey Swiader, Oriane Tasta, Frédéric Pont, Frédéric Rodriguez

Free Radic Biol Med· September 2019

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Selective Targeting of the Interconversion between Glucosylceramide and Ceramide by Scaffold Tailoring of Iminosugar Inhibitors.
Cécile Baudoin-Dehoux, Tessa Castellan, Frédéric Rodriguez, Arnaud Rives, Fabien Stauffert

Molecules· January 2019

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Iminosugar-based ceramide mimicry for the design of new CERT START domain ligands.
Cécile Santos, Fabien Stauffert, Stéphanie Ballereau, Cécile Dehoux, Frédéric Rodriguez

Bioorg Med Chem· March 2017

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Pyrrolidinone and pyrrolidine derivatives: Evaluation as inhibitors of InhA and Mycobacterium tuberculosis.
Tetiana Matviiuk, Jan Madacki, Giorgia Mori, Beatrice Silvia Orena, Christophe Menendez, Frédéric Rodriguez

Eur J Med Chem· November 2016

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Asymmetric Synthesis and Binding Study of New Long-Chain HPA-12 Analogues as Potent Ligands of the Ceramide Transfer Protein CERT.
Andrej Ďuriš, Adam Daïch, Cécile Santos, Laurence Fleury, Frédéric Ausseil, Frédéric Rodriguez

Chemistry· May 2016

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Hemisynthesis, Antitumoral Effect, and Molecular Docking Studies of Ferutinin and Its Analogues.
Rémi Safi, Fréderic Rodriguez, Georges Hilal, Mona Diab-Assaf, Youssef Diab

Chem Biol Drug Des· March 2016

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Design, synthesis and evaluation of new GEQ derivatives as inhibitors of InhA enzyme and Mycobacterium tuberculosis growth.
Aurélien Chollet, Giorgia Mori, Christophe Menendez, Frédéric Rodriguez, Isabelle Fabing

Eur J Med Chem· August 2015

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The CERT antagonist HPA-12: first practical synthesis and individual binding evaluation of the four stereoisomers.
Cécile Santos, Laurence Fleury, Frédéric Rodriguez, Jozef Markus, Dušan Berkeš

Bioorg Med Chem· May 2015

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Synthesis and in vitro antiproliferative activity of amido and amino analogues of the marine alkaloid isogranulatimide.
Hubert Lavrard, Béatrice Salvetti, Véronique Mathieu, Frédéric Rodriguez, Robert Kiss

ChemMedChem· April 2015

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Design, chemical synthesis of 3-(9H-fluoren-9-yl)pyrrolidine-2,5-dione derivatives and biological activity against enoyl-ACP reductase (InhA) and Mycobacterium tuberculosis.
Tetiana Matviiuk, Frédéric Rodriguez, Nathalie Saffon, Sonia Mallet-Ladeira, Marian Gorichko

Eur J Med Chem· September 2014

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Design of granulatimide and isogranulatimide analogues as potential Chk1 inhibitors: Study of amino-platforms for their synthesis.
Hubert Lavrard, Frédéric Rodriguez, Evelyne Delfourne

Bioorg Med Chem· September 2014

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Synthesis of 3-heteryl substituted pyrrolidine-2,5-diones via catalytic Michael reaction and evaluation of their inhibitory activity against InhA and Mycobacterium tuberculosis.
Tetiana Matviiuk, Giorgia Mori, Christian Lherbet, Frédéric Rodriguez, Maria Rosalia Pasca

Eur J Med Chem· January 2014

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Synthesis and evaluation of α-ketotriazoles and α,β-diketotriazoles as inhibitors of Mycobacterium tuberculosis.
Christophe Menendez, Frédéric Rodriguez, Ana Luisa de Jesus Lopes Ribeiro, Francesca Zara, Céline Frongia

Eur J Med Chem· November 2013

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