Publications by authors named "Jennifer Thomason"

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Discovery of novel N-hydroxy-2-arylisoindoline-4-carboxamides as potent and selective inhibitors of HDAC11.
Matthew W Martin, Jennifer Y Lee, David R Lancia, Pui Yee Ng, Bingsong Han, Jennifer R Thomason

Bioorg Med Chem Lett· July 2018

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Discovery of Clinical Candidate 1-{[(2S,3S,4S)-3-Ethyl-4-fluoro-5-oxopyrrolidin-2-yl]methoxy}-7-methoxyisoquinoline-6-carboxamide (PF-06650833), a Potent, Selective Inhibitor of Interleukin-1 Receptor Associated Kinase 4 (IRAK4), by Fragment-Based Drug Design.
Katherine L Lee, Catherine M Ambler, David R Anderson, Brian P Boscoe, Andrea G Bree, Jennifer R Thomason

J Med Chem· July 2017

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Discovery of isoquinolinone indole acetic acids as antagonists of chemoattractant receptor homologous molecule expressed on Th2 cells (CRTH2) for the treatment of allergic inflammatory diseases.
Neelu Kaila, Bruce Follows, Louis Leung, Jennifer Thomason, Adrian Huang

J Med Chem· February 2014

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Diazine indole acetic acids as potent, selective, and orally bioavailable antagonists of chemoattractant receptor homologous molecule expressed on Th2 cells (CRTH2) for the treatment of allergic inflammatory diseases.
Neelu Kaila, Adrian Huang, Alessandro Moretto, Bruce Follows, Kristin Janz, Jennifer Thomason

J Med Chem· June 2012

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Continued exploration of biphenylsulfonamide scaffold as a platform for aggrecanase-1 inhibition.
Yonghan Hu, Li Xing, Jennifer R Thomason, Jason Xiang, Manus Ipek

Bioorg Med Chem Lett· November 2011

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3,4-Disubstituted benzofuran P1' MMP-13 inhibitors: optimization of selectivity and reduction of protein binding.
Wei Li, Yonghan Hu, Jianchang Li, Jennifer R Thomason, Dianne DeVincentis

Bioorg Med Chem Lett· August 2009

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Synthesis and biological evaluation of ((4-keto)-phenoxy)methyl biphenyl-4-sulfonamides: a class of potent aggrecanase-1 inhibitors.
Darrin W Hopper, Matthew D Vera, David How, Joshua Sabatini, Jason S Xiang, Jennifer Thomason

Bioorg Med Chem Lett· May 2009

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Indole cytosolic phospholipase A2 alpha inhibitors: discovery and in vitro and in vivo characterization of 4-{3-[5-chloro-2-(2-{[(3,4-dichlorobenzyl)sulfonyl]amino}ethyl)-1-(diphenylmethyl)-1H-indol-3-yl]propyl}benzoic acid, efipladib.
John C McKew, Katherine L Lee, Marina W H Shen, Paresh Thakker, Megan A Foley, Jennifer Thomason

J Med Chem· June 2008

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Identification of a novel class of selective Tpl2 kinase inhibitors: 4-Alkylamino-[1,7]naphthyridine-3-carbonitriles.
Neelu Kaila, Neal Green, Huan-Qiu Li, Yonghan Hu, Kristin Janz, Jennifer Thomason

Bioorg Med Chem· October 2007

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Inhibitors of tumor progression loci-2 (Tpl2) kinase and tumor necrosis factor alpha (TNF-alpha) production: selectivity and in vivo antiinflammatory activity of novel 8-substituted-4-anilino-6-aminoquinoline-3-carbonitriles.
Neal Green, Yonghan Hu, Kristin Janz, Huan-Qiu Li, Neelu Kaila, Jennifer Thomason

J Med Chem· September 2007

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Inhibition of Tpl2 kinase and TNFalpha production with quinoline-3-carbonitriles for the treatment of rheumatoid arthritis.
Yonghan Hu, Neal Green, Lori K Gavrin, Kristin Janz, Neelu Kaila, Jennifer R Thomason

Bioorg Med Chem Lett· December 2006

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Synthesis and biological evaluation of biphenylsulfonamide carboxylate aggrecanase-1 inhibitors.
Jason S Xiang, Yonghan Hu, Thomas S Rush, Jennifer R Thomason, Manus Ipek

Bioorg Med Chem Lett· January 2006

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Inhibition of Tpl2 kinase and TNF-alpha production with 1,7-naphthyridine-3-carbonitriles: synthesis and structure-activity relationships.
Lori Krim Gavrin, Neal Green, Yonghan Hu, Kristin Janz, Neelu Kaila, Jennifer R Thomason

Bioorg Med Chem Lett· December 2005

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Potent, selective, and orally bioavailable matrix metalloproteinase-13 inhibitors for the treatment of osteoarthritis.
Yonghan Hu, Jason S Xiang, Martin J DiGrandi, Xuemei Du, Manus Ipek, Jennifer R Thomason

Bioorg Med Chem· December 2005

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Synthesis and SAR of highly selective MMP-13 inhibitors.
Jianchang Li, Thomas S Rush, Wei Li, Dianne DeVincentis, Xuemei Du, Jennifer R Thomason

Bioorg Med Chem Lett· November 2005

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