Publications by authors named "Marc Lecomte"

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PROTAC Enabling Formulation : Implications of the Polymeric Carrier Eudragit E PO.
Nicole Hofmann, Florian Johann, Katharina Krollik, Andreas Marx, Heide Marika Duevel, Marc Lecomte

Mol Pharm· October 2025

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and ADME of heterobifunctional degraders: a tailored approach to optimize DMPK properties of PROTACs©.
Christine Katharina Maurer, Zhizhou Fang, Christina Schindler, Gianna Pohl, Fouzia Machrouhi-Porcher, Marc Lecomte

RSC Med Chem· February 2025

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Dual A2A/A2B Adenosine Receptor Antagonist M1069 Counteracts Immunosuppressive Mechanisms of Adenosine and Reduces Tumor Growth In Vivo.
Kai Schiemann, Natalya Belousova, Armine Matevossian, Kalyan C Nallaparaju, Giorgio Kradjian, Marc Lecomte

Mol Cancer Ther· November 2024

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Discovery of Cycloalkyl[]thiophenes as Novel Scaffolds for Hypoxia-Inducible Factor-2α Inhibitors.
Hans-Peter Buchstaller, Ada Sala-Hojman, Matthias Leiendecker, Joachim Albers, Uwe Anlauf, Marc Lecomte

J Med Chem· July 2023

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Identification of solubility-limited absorption of oral anticancer drugs using PBPK modeling based on rat PK and its relevance to human.
Christina Fink, Marc Lecomte, Lassina Badolo, Knut Wagner, Karsten Mäder

Eur J Pharm Sci· September 2020

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Prediction of volume of distribution in humans: analysis of eight methods and their application in drug discovery.
Carl Petersson, Orestis Papasouliotis, Marc Lecomte, Lassina Badolo, Hugues Dolgos

Xenobiotica· March 2020

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Improved Prediction of in Vivo Supersaturation and Precipitation of Poorly Soluble Weakly Basic Drugs Using a Biorelevant Bicarbonate Buffer in a Gastrointestinal Transfer Model.
Christian Jede, Christian Wagner, Holger Kubas, Markus Weigandt, Christian Weber, Marc Lecomte

Mol Pharm· September 2019

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Structure-based design of 7-azaindole-pyrrolidine amides as inhibitors of 11β-hydroxysteroid dehydrogenase type I.
Eric Valeur, Serge Christmann-Franck, Franck Lepifre, Denis Carniato, Daniel Cravo, Marc Lecomte

Bioorg Med Chem Lett· September 2012

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Discovery and structure-guided drug design of inhibitors of 11beta-hydroxysteroid-dehydrogenase type I based on a spiro-carboxamide scaffold.
Franck Lepifre, Serge Christmann-Franck, Didier Roche, Caroline Leriche, Denis Carniato, Marc Lecomte

Bioorg Med Chem Lett· July 2009

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Discovery and structure-activity relationships of pentanedioic acid diamides as potent inhibitors of 11beta-hydroxysteroid dehydrogenase type I.
Didier Roche, Denis Carniato, Caroline Leriche, Franck Lepifre, Serge Christmann-Franck, Marc Lecomte

Bioorg Med Chem Lett· May 2009

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Involvement of caspase-10 in advanced glycation end-product-induced apoptosis of bovine retinal pericytes in culture.
Marc Lecomte, Ulriche Denis, Daniel Ruggiero, Michel Lagarde, Nicolas Wiernsperger

Biochim Biophys Acta· August 2004

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Advanced glycation end-products induce apoptosis of bovine retinal pericytes in culture: involvement of diacylglycerol/ceramide production and oxidative stress induction.
Ulriche Denis, Marc Lecomte, Clarisse Paget, Daniel Ruggiero, Nicolas Wiernsperger

Free Radic Biol Med· July 2002

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