Publications by authors named "Neil Garton"

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Bromodomain inhibitor i-BET858 triggers a unique transcriptional response coupled to enhanced DNA damage, cell cycle arrest and apoptosis in high-grade ovarian carcinoma cells.
Marcos Quintela, David W James, Agne Pociute, Lydia Powell, Kadie Edwards, Neil Garton

Clin Epigenetics· April 2023

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Click chemistry enables preclinical evaluation of targeted epigenetic therapies.
Dean S Tyler, Johanna Vappiani, Tatiana Cañeque, Enid Y N Lam, Aoife Ward, Neil Garton

Science· June 2017

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Optimisation of a novel series of potent and orally bioavailable azanaphthyridine SYK inhibitors.
Neil S Garton, Michael D Barker, Rob P Davis, Clement Douault, Edward Hooper-Greenhill

Bioorg Med Chem Lett· October 2016

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Interrogating the Druggability of the 2-Oxoglutarate-Dependent Dioxygenase Target Class by Chemical Proteomics.
Gérard Joberty, Markus Boesche, Jack A Brown, Dirk Eberhard, Neil S Garton

ACS Chem Biol· July 2016

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Functional interdependence of BRD4 and DOT1L in MLL leukemia.
Omer Gilan, Enid Y N Lam, Isabelle Becher, Dave Lugo, Ester Cannizzaro, Neil Garton

Nat Struct Mol Biol· July 2016

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Cell Penetrant Inhibitors of the KDM4 and KDM5 Families of Histone Lysine Demethylases. 2. Pyrido[3,4-d]pyrimidin-4(3H)-one Derivatives.
Susan M Westaway, Alex G S Preston, Michael D Barker, Fiona Brown, Jack A Brown, Neil Garton

J Med Chem· February 2016

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Autism-like syndrome is induced by pharmacological suppression of BET proteins in young mice.
Josefa M Sullivan, Ana Badimon, Uwe Schaefer, Pinar Ayata, James Gray, Neil Garton

J Exp Med· October 2015

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Discovery of GSK143, a highly potent, selective and orally efficacious spleen tyrosine kinase inhibitor.
John Liddle, Francis L Atkinson, Michael D Barker, Paul S Carter, Neil R Curtis, Neil S Garton

Bioorg Med Chem Lett· October 2011

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Discovery of biaryl inhibitors of H+/K+ ATPase.
Neil Garton, Nick Bailey, Mark Bamford, Emmanuel Demont, Irene Farre-Gutierrez

Bioorg Med Chem Lett· February 2010

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Evaluation of basic, heterocyclic ring systems as templates for use as potassium competitive acid blockers (pCABs).
Terry Panchal, Nick Bailey, Mark Bamford, Emmanuel Demont, Richard Elliott, Neil Garton

Bioorg Med Chem Lett· December 2009

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Orally active C-6 heteroaryl- and heterocyclyl-substituted imidazo[1,2-a]pyridine acid pump antagonists (APAs).
Nick Bailey, Mark J Bamford, Delphine Brissy, Joanna Brookfield, Emmanuel Demont, Neil Garton

Bioorg Med Chem Lett· July 2009

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Pyridone derivatives as potent, orally bioavailable VLA-4 integrin antagonists.
Jason Witherington, Emma L Blaney, Vincent Bordas, Richard L Elliott, Alessandra Gaiba, Neil Garton

Bioorg Med Chem Lett· November 2006

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6-aryl-pyrazolo[3,4-b]pyridines: potent inhibitors of glycogen synthase kinase-3 (GSK-3).
Jason Witherington, Vincent Bordas, Alessandra Gaiba, Neil S Garton, Antoinette Naylor

Bioorg Med Chem Lett· September 2003

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