Publications by authors named "Neil Norcross"

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lysyl-tRNA synthetase inhibitors define the interplay between solubility and permeability required to achieve efficacy.
Nicola Caldwell, Caroline Peet, Peter Miller, Beatrice L Colon, Malcolm G Taylor, Neil R Norcross

Sci Transl Med· October 2024

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Sperm Toolbox-A selection of small molecules to study human spermatozoa.
Franz S Gruber, Anthony Richardson, Zoe C Johnston, Rachel Myles, Neil R Norcross

PLoS One· February 2024

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Identification and Optimization of Novel Inhibitors of the Polyketide Synthase 13 Thioesterase Domain with Antitubercular Activity.
Simon R Green, Caroline Wilson, Thomas C Eadsforth, Avinash S Punekar, Fabio K Tamaki, Neil R Norcross

J Med Chem· November 2023

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Male contraceptive development: A medicinal chemistry perspective.
Neil R Norcross, Irene Georgiou, Zoe C Johnston, Franz S Gruber, Jason R Swedlow

Eur J Med Chem· December 2022

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Compounds enhancing human sperm motility identified using a high-throughput phenotypic screening platform.
Franz S Gruber, Zoe C Johnston, Neil R Norcross, Irene Georgiou, Caroline Wilson

Hum Reprod· March 2022

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High-throughput phenotypic screening of the human spermatozoon.
Zoe C Johnston, Franz S Gruber, Sean G Brown, Neil R Norcross, Jason Swedlow

Reproduction· December 2021

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Substituted Aminoacetamides as Novel Leads for Malaria Treatment.
Neil R Norcross, Caroline Wilson, Beatriz Baragaña, Irene Hallyburton, Maria Osuna-Cabello

ChemMedChem· July 2019

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Lysyl-tRNA synthetase as a drug target in malaria and cryptosporidiosis.
Beatriz Baragaña, Barbara Forte, Ryan Choi, Stephen Nakazawa Hewitt, Juan A Bueren-Calabuig, Neil R Norcross

Proc Natl Acad Sci U S A· April 2019

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Discovery of a Quinoline-4-carboxamide Derivative with a Novel Mechanism of Action, Multistage Antimalarial Activity, and Potent in Vivo Efficacy.
Beatriz Baragaña, Neil R Norcross, Caroline Wilson, Achim Porzelle, Irene Hallyburton

J Med Chem· November 2016

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Corrigendum: A novel multiple-stage antimalarial agent that inhibits protein synthesis.
Beatriz Baragaña, Irene Hallyburton, Marcus C S Lee, Neil R Norcross, Raffaella Grimaldi

Nature· September 2016

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Trisubstituted Pyrimidines as Efficacious and Fast-Acting Antimalarials.
Neil R Norcross, Beatriz Baragaña, Caroline Wilson, Irene Hallyburton, Maria Osuna-Cabello

J Med Chem· July 2016

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Validation of N-myristoyltransferase as Potential Chemotherapeutic Target in Mammal-Dwelling Stages of Trypanosoma cruzi.
Linda J Herrera, Stephen Brand, Andres Santos, Lilian L Nohara, Justin Harrison, Neil R Norcross

PLoS Negl Trop Dis· April 2016

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Discovery of Inhibitors of Trypanosoma brucei by Phenotypic Screening of a Focused Protein Kinase Library.
Andrew Woodland, Stephen Thompson, Laura A T Cleghorn, Neil Norcross, Manu De Rycker

ChemMedChem· November 2015

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A novel multiple-stage antimalarial agent that inhibits protein synthesis.
Beatriz Baragaña, Irene Hallyburton, Marcus C S Lee, Neil R Norcross, Raffaella Grimaldi

Nature· June 2015

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Lead optimization of a pyrazole sulfonamide series of Trypanosoma brucei N-myristoyltransferase inhibitors: identification and evaluation of CNS penetrant compounds as potential treatments for stage 2 human African trypanosomiasis.
Stephen Brand, Neil R Norcross, Stephen Thompson, Justin R Harrison, Victoria C Smith

J Med Chem· December 2014

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Exploring the Trypanosoma brucei Hsp83 potential as a target for structure guided drug design.
Juan Carlos Pizarro, Tanya Hills, Guillermo Senisterra, Amy K Wernimont, Claire Mackenzie, Neil R Norcross

PLoS Negl Trop Dis· May 2014

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Substituted 2-phenylimidazopyridines: a new class of drug leads for human African trypanosomiasis.
Hari Babu Tatipaka, J Robert Gillespie, Arnab K Chatterjee, Neil R Norcross, Matthew A Hulverson

J Med Chem· February 2014

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Dialkylimidazole inhibitors of Trypanosoma cruzi sterol 14α-demethylase as anti-Chagas disease agents.
Praveen Kumar Suryadevara, Kishore Kumar Racherla, Srinivas Olepu, Neil R Norcross, Hari Babu Tatipaka

Bioorg Med Chem Lett· December 2013

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Discovery of a novel class of orally active trypanocidal N-myristoyltransferase inhibitors.
Stephen Brand, Laura A T Cleghorn, Stuart P McElroy, David A Robinson, Victoria C Smith, Neil R Norcross

J Med Chem· January 2012

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Identification of inhibitors of the Leishmania cdc2-related protein kinase CRK3.
Laura A T Cleghorn, Andrew Woodland, Iain T Collie, Leah S Torrie, Neil Norcross

ChemMedChem· December 2011

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Total synthesis of (+/-)-alpha-isosparteine, (+/-)-beta-isosparteine, and (+/-)-sparteine from a common tetraoxobispidine intermediate.
Neil R Norcross, John P Melbardis, Margarita Ferris Solera, Mark A Sephton, Colin Kilner

J Org Chem· October 2008

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A practical synthesis of (+/-)-alpha-isosparteine from a tetraoxobispidine core.
Paul R Blakemore, Colin Kilner, Neil R Norcross, Peter C Astles

Org Lett· October 2005

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