Publications by authors named "Roberto Perrone"

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Deciphering the Supramolecular Organization of Multiple Guests Inside a Microporous MOF to Understand their Release Profile.
Davide Balestri, Paolo P Mazzeo, Roberto Perrone, Fabio Fornari, Federica Bianchi

Angew Chem Int Ed Engl· April 2021

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Why PB28 Could Be a Covid 2019 Game Changer?
Nicola Antonio Colabufo, Marcello Leopoldo, Savina Ferorelli, Carmen Abate, Marialessandra Contino, Maria Grazia Perrone, Roberto Perrone

ACS Med Chem Lett· October 2020

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An innovative small molecule for promoting neuroreparative strategies.
Nicola Antonio Colabufo, Marialessandra Contino, Mariangela Cantore, Francesco Berardi, Roberto Perrone

RSC Adv· January 2018

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Design and Synthesis of New Selective P-gp Substrates and Inhibitors.
Mariangela Cantore, Marcello Leopoldo, Francesco Berardi, Roberto Perrone, Nicola Antonio Colabufo

Curr Pharm Des· December 2017

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Novel ureidopropanamide based N-formyl peptide receptor 2 (FPR2) agonists with potential application for central nervous system disorders characterized by neuroinflammation.
Madia Letizia Stama, Joanna Ślusarczyk, Enza Lacivita, Liliya N Kirpotina, Igor A Schepetkin, Roberto Perrone

Eur J Med Chem· December 2017

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Functional N-Formyl Peptide Receptor 2 (FPR2) Antagonists Based on the Ureidopropanamide Scaffold Have Potential To Protect Against Inflammation-Associated Oxidative Stress.
Madia L Stama, Enza Lacivita, Liliya N Kirpotina, Mauro Niso, Roberto Perrone

ChemMedChem· November 2017

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Targets for Drug Therapy for Autism Spectrum Disorder: Challenges and Future Directions.
Enza Lacivita, Roberto Perrone, Lucia Margari, Marcello Leopoldo

J Med Chem· November 2017

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Structure-activity relationship study towards non-peptidic positron emission tomography (PET) radiotracer for gastrin releasing peptide receptors: Development of [F] (S)-3-(1H-indol-3-yl)-N-[1-[5-(2-fluoroethoxy)pyridin-2-yl]cyclohexylmethyl]-2-methyl-2-[3-(4-nitrophenyl)ureido]propionamide.
Enza Lacivita, Ermelinda Lucente, Chantal Kwizera, Ines F Antunes, Mauro Niso, Roberto Perrone

Bioorg Med Chem· January 2017

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Structural modifications of the serotonin 5-HT7 receptor agonist N-(4-cyanophenylmethyl)-4-(2-biphenyl)-1-piperazinehexanamide (LP-211) to improve in vitro microsomal stability: A case study.
Enza Lacivita, Sabina Podlewska, Luisa Speranza, Mauro Niso, Grzegorz Satała, Roberto Perrone, Carla Perrone-Capano

Eur J Med Chem· September 2016

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Radiosynthesis and in vivo Evaluation of Carbon-11 (2S)-3-(1H-Indol-3-yl)-2-{[(4-methoxyphenyl)carbamoyl]amino}-N-{[1-(5-methoxypyridin-2-yl)cyclohexyl]methyl}propanamide: An Attempt to Visualize Brain Formyl Peptide Receptors in Mouse Models of Neuroinflammation.
Enza Lacivita, Madia Letizia Stama, Jun Maeda, Masayuki Fujinaga, Akiko Hatori, Roberto Perrone

Chem Biodivers· July 2016

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Functionalized Coumarine Fragment to Obtain Fluorescent and Selective P-Glycoprotein Ligands.
Elena Capparelli, Marialessandra Contino, Maria G Perrone, Francesco Berardi, Roberto Perrone

Arch Pharm (Weinheim)· March 2016

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Arylpiperazine agonists of the serotonin 5-HT1A receptor preferentially activate cAMP signaling versus recruitment of β-arrestin-2.
Nikolas Stroth, Mauro Niso, Nicola A Colabufo, Roberto Perrone, Per Svenningsson

Bioorg Med Chem· August 2015

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Novel 3-(1H-indol-3-yl)-2-[3-(4-methoxyphenyl)ureido]propanamides as selective agonists of human formyl-peptide receptor 2.
Enza Lacivita, Igor A Schepetkin, Madia L Stama, Liliya N Kirpotina, Nicola A Colabufo, Roberto Perrone

Bioorg Med Chem· July 2015

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From mixed sigma-2 receptor/P-glycoprotein targeting agents to selective P-glycoprotein modulators: small structural changes address the mechanism of interaction at the efflux pump.
Carmen Abate, Maria Laura Pati, Marialessandra Contino, Nicola Antonio Colabufo, Roberto Perrone

Eur J Med Chem· January 2015

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SAR studies on tetrahydroisoquinoline derivatives: the role of flexibility and bioisosterism to raise potency and selectivity toward P-glycoprotein.
Elena Capparelli, Laura Zinzi, Mariangela Cantore, Marialessandra Contino, Maria Grazia Perrone, Roberto Perrone

J Med Chem· December 2014

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Selective agonists for serotonin 7 (5-HT7) receptor and their applications in preclinical models: an overview.
Pantaleo Di Pilato, Mauro Niso, Walter Adriani, Emilia Romano, Domenica Travaglini, Roberto Perrone

Rev Neurosci· September 2014

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Trimethoxybenzanilide-based P-glycoprotein modulators: an interesting case of lipophilicity tuning by intramolecular hydrogen bonding.
Piero Tardia, Angela Stefanachi, Mauro Niso, Diana Antonella Stolfa, Giuseppe Felice Mangiatordi, Roberto Perrone

J Med Chem· August 2014

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Synthesis, radiolabeling and in vivo evaluation of [(11)C](R)-1-[4-[2-(4-methoxyphenyl)phenyl]piperazin-1-yl]-3-(2-pyrazinyloxy)-2-propanol, a potential PET radioligand for the 5-HT(7) receptor.
Hanne D Hansen, Enza Lacivita, Pantaleo Di Pilato, Matthias M Herth, Szabolcs Lehel, Roberto Perrone

Eur J Med Chem· May 2014

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SAR study on arylmethyloxyphenyl scaffold: looking for a P-gp nanomolar affinity.
Giulia Nesi, Nicola Antonio Colabufo, Marialessandra Contino, Maria Grazia Perrone, Maria Digiacomo, Roberto Perrone

Eur J Med Chem· April 2014

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Novel derivatives of 1-cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperazine (PB28) with improved fluorescent and σ receptors binding properties.
Carmen Abate, Mauro Niso, Roberta Marottoli, Chiara Riganti, Dario Ghigo, Roberto Perrone

J Med Chem· April 2014

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Design, synthesis, radiolabeling and in vivo evaluation of potential positron emission tomography (PET) radioligands for brain imaging of the 5-HT₇ receptor.
Enza Lacivita, Mauro Niso, Hanne D Hansen, Pantaleo Di Pilato, Matthias M Herth, Roberto Perrone

Bioorg Med Chem· March 2014

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Design, synthesis, lipophilic properties, and binding affinities of potential ligands in positron emission tomography (PET) for visualization of brain dopamine D4 receptors.
Enza Lacivita, Paola De Giorgio, Nicola A Colabufo, Francesco Berardi, Roberto Perrone

Chem Biodivers· February 2014

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PET radiotracers for imaging P-glycoprotein: the challenge for early diagnosis in AD.
Marcello Leopoldo, Marialessandra Contino, Francesco Berardi, Roberto Perrone, Nicola Antonio Colabufo

ChemMedChem· January 2014

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Sigma-2 receptor agonists as possible antitumor agents in resistant tumors: hints for collateral sensitivity.
Mauro Niso, Carmen Abate, Marialessandra Contino, Savina Ferorelli, Amalia Azzariti, Roberto Perrone

ChemMedChem· December 2013

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Development of 3,4-dihydroisoquinolin-1(2H)-one derivatives for the Positron Emission Tomography (PET) imaging of σ₂ receptors.
Carmen Abate, Svetlana V Selivanova, Adrienne Müller, Stefanie D Krämer, Roger Schibli, Roberto Perrone

Eur J Med Chem· November 2013

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