Publications by authors named "Stacie Bulfer"

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Discovery of vimseltinib (DCC-3014), a highly selective CSF1R switch-control kinase inhibitor, in clinical development for the treatment of Tenosynovial Giant Cell Tumor (TGCT).
Timothy M Caldwell, Yu Mi Ahn, Stacie L Bulfer, Cynthia B Leary, Molly M Hood

Bioorg Med Chem Lett· October 2022

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Discovery of acyl ureas as highly selective small molecule CSF1R kinase inhibitors.
Timothy M Caldwell, Michael D Kaufman, Scott C Wise, Yu Mi Ahn, Molly M Hood, Stacie L Bulfer

Bioorg Med Chem Lett· October 2022

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Ripretinib (DCC-2618) Is a Switch Control Kinase Inhibitor of a Broad Spectrum of Oncogenic and Drug-Resistant KIT and PDGFRA Variants.
Bryan D Smith, Michael D Kaufman, Wei-Ping Lu, Anu Gupta, Cynthia B Leary, Stacie L Bulfer

Cancer Cell· May 2019

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Optimization of Phenyl Indole Inhibitors of the AAA+ ATPase p97.
Matthew G LaPorte, James C Burnett, Raffaele Colombo, Stacie L Bulfer, Celeste Alverez

ACS Med Chem Lett· November 2018

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A threonine turnstile defines a dynamic amphiphilic binding motif in the AAA ATPase p97 allosteric binding site.
James C Burnett, Chaemin Lim, Brian D Peyser, Lalith P Samankumara, Marina Kovaliov, Stacie L Bulfer

Org Biomol Chem· May 2017

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p97 Disease Mutations Modulate Nucleotide-Induced Conformation to Alter Protein-Protein Interactions.
Stacie L Bulfer, Tsui-Fen Chou, Michelle R Arkin

ACS Chem Biol· August 2016

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2.3 Å resolution cryo-EM structure of human p97 and mechanism of allosteric inhibition.
Soojay Banerjee, Alberto Bartesaghi, Alan Merk, Prashant Rao, Stacie L Bulfer

Science· February 2016

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Allosteric Indole Amide Inhibitors of p97: Identification of a Novel Probe of the Ubiquitin Pathway.
Celeste Alverez, Stacie L Bulfer, Ramappa Chakrasali, Michael S Chimenti, Raymond J Deshaies

ACS Med Chem Lett· February 2016

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Structure-Activity Study of Bioisosteric Trifluoromethyl and Pentafluorosulfanyl Indole Inhibitors of the AAA ATPase p97.
Celeste Alverez, Michelle R Arkin, Stacie L Bulfer, Raffaele Colombo, Marina Kovaliov

ACS Med Chem Lett· December 2015

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A Fragment-Based Ligand Screen Against Part of a Large Protein Machine: The ND1 Domains of the AAA+ ATPase p97/VCP.
Michael S Chimenti, Stacie L Bulfer, R Jeffrey Neitz, Adam R Renslo, Matthew P Jacobson

J Biomol Screen· July 2015

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Altered cofactor regulation with disease-associated p97/VCP mutations.
Xiaoyi Zhang, Lin Gui, Xiaoyan Zhang, Stacie L Bulfer, Valentina Sanghez

Proc Natl Acad Sci U S A· April 2015

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Specific inhibition of p97/VCP ATPase and kinetic analysis demonstrate interaction between D1 and D2 ATPase domains.
Tsui-Fen Chou, Stacie L Bulfer, Conrad C Weihl, Kelin Li, Lev G Lis

J Mol Biol· July 2014

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Crystal structure of Saccharomyces cerevisiae Aro8, a putative α-aminoadipate aminotransferase.
Stacie L Bulfer, Joseph S Brunzelle, Raymond C Trievel

Protein Sci· October 2013

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Crystal structure of homoisocitrate dehydrogenase from Schizosaccharomyces pombe.
Stacie L Bulfer, Jenna M Hendershot, Raymond C Trievel

Proteins· February 2012

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Application of a high-throughput fluorescent acetyltransferase assay to identify inhibitors of homocitrate synthase.
Stacie L Bulfer, Thomas J McQuade, Martha J Larsen, Raymond C Trievel

Anal Biochem· March 2011

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Structural basis for L-lysine feedback inhibition of homocitrate synthase.
Stacie L Bulfer, Erin M Scott, Lorraine Pillus, Raymond C Trievel

J Biol Chem· April 2010

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Crystal structure and functional analysis of homocitrate synthase, an essential enzyme in lysine biosynthesis.
Stacie L Bulfer, Erin M Scott, Jean-François Couture, Lorraine Pillus, Raymond C Trievel

J Biol Chem· December 2009

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A coupled fluorescent assay for histone methyltransferases.
Evys Collazo, Jean-François Couture, Stacie Bulfer, Raymond C Trievel

Anal Biochem· July 2005

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