Publications by authors named "Azriel Schmidt"

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A novel selective androgen receptor modulator (SARM) MK-4541 exerts anti-androgenic activity in the prostate cancer xenograft R-3327G and anabolic activity on skeletal muscle mass & function in castrated mice.
Michael J Chisamore, Michael A Gentile, Gregory Michael Dillon, Matthew Baran, Carlo Gambone, Azriel Schmidt

J Steroid Biochem Mol Biol· October 2016

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Identification of an anabolic selective androgen receptor modulator that actively induces death of androgen-independent prostate cancer cells.
Azriel Schmidt, Robert S Meissner, Michael A Gentile, Michael J Chisamore, Evan E Opas

J Steroid Biochem Mol Biol· September 2014

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The preclinical efficacy, selectivity and pharmacologic profile of MK-5932, an insulin-sparing selective glucocorticoid receptor modulator.
Philip E Brandish, Kenneth Anderson, Gretchen A Baltus, Chang Bai, Christopher J Bungard, Azriel Schmidt

Eur J Pharmacol· February 2014

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Discovery of selective glucocorticoid receptor modulator MK-5932.
Christopher J Bungard, George D Hartman, Jesse J Manikowski, James J Perkins, Chang Bai, Azriel Schmidt

Bioorg Med Chem· December 2011

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Discovery of the selective androgen receptor modulator MK-0773 using a rational development strategy based on differential transcriptional requirements for androgenic anabolism versus reproductive physiology.
Azriel Schmidt, Donald B Kimmel, Chang Bai, Angela Scafonas, Sujane Rutledge

J Biol Chem· May 2010

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Identification of anabolic selective androgen receptor modulators with reduced activities in reproductive tissues and sebaceous glands.
Azriel Schmidt, Shun-Ichi Harada, Donald B Kimmel, Chang Bai, Fang Chen

J Biol Chem· December 2009

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Control of rat tail skin temperature regulation by estrogen receptor-beta selective ligand.
Evan E Opas, Angela Scafonas, Pascale V Nantermet, Robert R Wilkening, Elizabeth T Birzin, Azriel Schmidt

Maturitas· September 2009

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Design, synthesis, and biological evaluation of 16-substituted 4-azasteroids as tissue-selective androgen receptor modulators (SARMs).
Helen J Mitchell, William P Dankulich, George D Hartman, Thomayant Prueksaritanont, Azriel Schmidt

J Med Chem· August 2009

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Agonist-like SERM effects on ERalpha-mediated repression of MMP1 promoter activity predict in vivo effects on bone and uterus.
Angela Scafonas, Alfred A Reszka, Donald B Kimmel, Xiaoli Shirley Hou, Qin Su, Azriel Schmidt

J Steroid Biochem Mol Biol· June 2008

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Opportunities for development of novel therapies targeting steroid hormone receptors.
Chang Bai, Osvaldo Flores, Azriel Schmidt

Expert Opin Drug Discov· May 2007

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Antagonist-induced, activation function-2-independent estrogen receptor alpha phosphorylation.
Lorraine Lipfert, John E Fisher, Nan Wei, Angela Scafonas, Qin Su, Azriel Schmidt

Mol Endocrinol· March 2006

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Estrogenic control of thermoregulation in ERalphaKO and ERbetaKO mice.
Evan E Opas, Michael A Gentile, Donald B Kimmel, Gideon A Rodan, Azriel Schmidt

Maturitas· January 2006

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Direct agonist/antagonist functions of dehydroepiandrosterone.
Fang Chen, Kristin Knecht, Elizabeth Birzin, John Fisher, Hilary Wilkinson, Azriel Schmidt

Endocrinology· November 2005

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Interaction between the androgen receptor and RNase L mediates a cross-talk between the interferon and androgen signaling pathways.
David J Bettoun, Angela Scafonas, Su Jane Rutledge, Paul Hodor, Oliver Chen, Azriel Schmidt

J Biol Chem· November 2005

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Cross-talk between an activator of nuclear receptors-mediated transcription and the D1 dopamine receptor signaling pathway.
Azriel Schmidt, Robert Vogel, Su Jane Rutledge, Evan E Opas, Gideon A Rodan

Pharmacol Biochem Behav· March 2005

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Androgenic induction of growth and differentiation in the rodent uterus involves the modulation of estrogen-regulated genetic pathways.
Pascale V Nantermet, Patricia Masarachia, Michael A Gentile, Brenda Pennypacker, Jian Xu, Azriel Schmidt

Endocrinology· February 2005

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The LATS2/KPM tumor suppressor is a negative regulator of the androgen receptor.
Mark Powzaniuk, Sheila McElwee-Witmer, Robert L Vogel, Tadashi Hayami, Su Jane Rutledge, Azriel Schmidt

Mol Endocrinol· August 2004

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Rat tail skin temperature regulation by estrogen, phytoestrogens and tamoxifen.
Evan E Opas, Su Jane Rutledge, Robert L Vogel, Gideon A Rodan, Azriel Schmidt

Maturitas· August 2004

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Steroid hormone receptors and drug discovery: therapeutic opportunities and assay designs.
Chang Bai, Azriel Schmidt, Leonard P Freedman

Assay Drug Dev Technol· December 2003

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A novel liver X receptor agonist establishes species differences in the regulation of cholesterol 7alpha-hydroxylase (CYP7a).
John G Menke, Karen L Macnaul, Nancy S Hayes, Joanne Baffic, Yu-Sheng Chao, Azriel Schmidt

Endocrinology· July 2002

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