Publications by authors named "Jon E Hawkinson"

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Macrocyclic dihydropyridine analogs as pan-BET BD2-preferred inhibitors.
Jiewei Jiang, Taimeng Liang, Jonathan Solberg, Alice Chan, Prakriti Kalra, Jon E Hawkinson

Eur J Med Chem· June 2025

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Strategies for developing retinoic acid receptor alpha-selective antagonists as novel agents for male contraception.
Md Abdullah Al Noman, Rebecca A D Cuellar, Jillian L Kyzer, Sanny S W Chung, Narsihmulu Cheryala, Jon E Hawkinson

Eur J Med Chem· December 2023

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Investigation of selective retinoic acid receptor alpha antagonist ER-50891 and related analogs for male contraception.
Jillian L Kyzer, Md Abdullah Al Noman, Rebecca A D Cuellar, Sanny S W Chung, Soma Maitra, Jon E Hawkinson

Arch Pharm (Weinheim)· July 2023

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Development of allosteric and selective CDK2 inhibitors for contraception with negative cooperativity to cyclin binding.
Erik B Faber, Luxin Sun, Jian Tang, Emily Roberts, Sornakala Ganeshkumar, Jon E Hawkinson

Nat Commun· June 2023

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Screening through Lead Optimization of High Affinity, Allosteric Cyclin-Dependent Kinase 2 (CDK2) Inhibitors as Male Contraceptives That Reduce Sperm Counts in Mice.
Erik B Faber, Nan Wang, Kristen John, Luxin Sun, Henry L Wong, Jon E Hawkinson

J Med Chem· February 2023

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Corrigendum: Discovery and Characterization of Multiple Classes of Human CatSper Blockers.
Erick J Carlson, Rawle Francis, Yutong Liu, Ping Li, Maximilian Lyon, Jon E Hawkinson

ChemMedChem· October 2022

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Discovery and Characterization of Multiple Classes of Human CatSper Blockers.
Erick J Carlson, Rawle Francis, Yutong Liu, Ping Li, Maximilian Lyon, Jon E Hawkinson

ChemMedChem· August 2022

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Steroidal Antagonists of Progesterone- and Prostaglandin E-Induced Activation of the Cation Channel of Sperm.
Erick J Carlson, Gunda I Georg, Jon E Hawkinson

Mol Pharmacol· January 2022

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FBNTI, a DOR-Selective Antagonist That Allosterically Activates MOR within a MOR-DOR Heteromer.
Eyup Akgün, Mary M Lunzer, Defeng Tian, Michael Ansonoff, John Pintar, Jon E Hawkinson

Biochemistry· May 2021

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Quantifying the Selectivity of Protein-Protein and Small Molecule Interactions with Fluorinated Tandem Bromodomain Reader Proteins.
Prakriti Kalra, Logan McGraw, Jennifer R Kimbrough, Anil K Pandey, Jonathan Solberg, Jon E Hawkinson

ACS Chem Biol· November 2020

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Development of WEE2 kinase inhibitors as novel non-hormonal female contraceptives that target meiosis†.
Carol B Hanna, Deepti Mudaliar, Kristen John, C Leigh Allen, Luxin Sun, Jon E Hawkinson

Biol Reprod· August 2020

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Cooperativity Between Orthosteric Inhibitors and Allosteric Inhibitor 8-Anilino-1-Naphthalene Sulfonic Acid (ANS) in Cyclin-Dependent Kinase 2.
Erik B Faber, Defeng Tian, David Burban, Nicholas M Levinson, Jon E Hawkinson

ACS Chem Biol· July 2020

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Automated Live-Cell Imaging of Synapses in Rat and Human Neuronal Cultures.
Matthew V Green, Thomas Pengo, Jonathan D Raybuck, Tahmina Naqvi, Hannah M McMullan, Jon E Hawkinson

Front Cell Neurosci· October 2019

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The anti-parasitic agent suramin and several of its analogues are inhibitors of the DNA binding protein Mcm10.
Carolyn N Paulson, Kristen John, Ryan M Baxley, Fredy Kurniawan, Kayo Orellana, Jon E Hawkinson

Open Biol· August 2019

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7-Methylation of Chenodeoxycholic Acid Derivatives Yields a Substantial Increase in TGR5 Receptor Potency.
Ali Nakhi, Connor M McDermott, Kristen L Stoltz, Kristen John, Jon E Hawkinson

J Med Chem· July 2019

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Design, Synthesis, and Characterization of a Fluorescence Polarization Pan-BET Bromodomain Probe.
Carolyn N Paulson, Xianghong Guan, Alex M Ayoub, Alice Chan, Rezaul M Karim, Jon E Hawkinson

ACS Med Chem Lett· December 2018

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Reduction of protein kinase A-mediated phosphorylation of ATXN1-S776 in Purkinje cells delays onset of Ataxia in a SCA1 mouse model.
Judit M Pérez Ortiz, Nissa Mollema, Nicholas Toker, Carolyn J Adamski, Brennon O'Callaghan, Jon E Hawkinson

Neurobiol Dis· August 2018

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Design, Synthesis, and in Vitro and in Vivo Evaluation of Ouabain Analogues as Potent and Selective Na,K-ATPase α4 Isoform Inhibitors for Male Contraception.
Shameem Sultana Syeda, Gladis Sánchez, Kwon Ho Hong, Jon E Hawkinson, Gunda I Georg

J Med Chem· March 2018

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Potent Pyrimidine and Pyrrolopyrimidine Inhibitors of Testis-Specific Serine/Threonine Kinase 2 (TSSK2).
Jon E Hawkinson, Rondedrick Sinville, Deepti Mudaliar, Jagathpala Shetty, Timothy Ward

ChemMedChem· November 2017

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Recombinant production of enzymatically active male contraceptive drug target hTSSK2 - Localization of the TSKS domain phosphorylated by TSSK2.
Jagathpala Shetty, Rondedrick Sinville, Igor A Shumilin, Wladek Minor, Jianhai Zhang, Jon E Hawkinson

Protein Expr Purif· May 2016

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Human Adenine Nucleotide Translocase (ANT) Modulators Identified by High-Throughput Screening of Transgenic Yeast.
Yujian Zhang, Defeng Tian, Hironori Matsuyama, Takashi Hamazaki, Takayuki Shiratsuchi, Jon E Hawkinson

J Biomol Screen· April 2016

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The Fungal Sexual Pheromone Sirenin Activates the Human CatSper Channel Complex.
Shameem Sultana Syeda, Erick J Carlson, Melissa R Miller, Rawle Francis, David E Clapham, Jon E Hawkinson

ACS Chem Biol· February 2016

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Probing the S2' Subsite of the Anthrax Toxin Lethal Factor Using Novel N-Alkylated Hydroxamates.
Elbek K Kurbanov, Ting-Lan Chiu, Jonathan Solberg, Subhashree Francis, Kimberly M Maize, Jon E Hawkinson

J Med Chem· November 2015

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From HTS to Phase I: the Institute for Therapeutics Discovery and Development at the University of Minnesota.
Peter I Dosa, Gunda I Georg, Vadim J Gurvich, Jon E Hawkinson, Michael A Walters

Comb Chem High Throughput Screen· March 2014

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Quantification of adverse events associated with functional MRI scanning and with real-time fMRI-based training.
Jon E Hawkinson, Amy J Ross, Sudharshan Parthasarathy, David J Scott, Ella A Laramee

Int J Behav Med· September 2012

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