Publications by authors named "Marc Labelle"

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Characterization of a KDM5 small molecule inhibitor with antiviral activity against hepatitis B virus.
Sarah A Gilmore, Danny Tam, Tara L Cheung, Chelsea Snyder, Julie Farand, Marc Labelle

PLoS One· December 2022

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Inhibition of demethylases by GSK-J1/J4.
Bo Heinemann, Jesper Morten Nielsen, Heidi Rye Hudlebusch, Michael J Lees, Dorthe Vang Larsen, Marc Labelle

Nature· October 2014

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Discovery of 6-phenylpyrimido[4,5-b][1,4]oxazines as potent and selective acyl CoA:diacylglycerol acyltransferase 1 (DGAT1) inhibitors with in vivo efficacy in rodents.
Brian M Fox, Kazuyuki Sugimoto, Kiyosei Iio, Atsuhito Yoshida, Jian Ken Zhang, Marc Labelle

J Med Chem· April 2014

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Discovery and optimization of a series of liver X receptor antagonists.
XianYun Jiao, David J Kopecky, Ben Fisher, Derek E Piper, Marc Labelle

Bioorg Med Chem Lett· September 2012

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Discovery of a new binding mode for a series of liver X receptor agonists.
David J Kopecky, Xian Yun Jiao, Ben Fisher, Sharon McKendry, Marc Labelle

Bioorg Med Chem Lett· April 2012

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A novel series of IKKβ inhibitors part II: description of a potent and pharmacologically active series of analogs.
Timothy D Cushing, Vijay Baichwal, Karen Berry, Roland Billedeau, Viola Bordunov, Marc Labelle

Bioorg Med Chem Lett· January 2011

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A novel series of IKKβ inhibitors part I: Initial SAR studies of a HTS hit.
Timothy D Cushing, Vijay Baichwal, Karen Berry, Roland Billedeau, Viola Bordunov, Marc Labelle

Bioorg Med Chem Lett· January 2011

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The synthesis and SAR of novel diarylsulfone 11β-HSD1 inhibitors.
Xuelei Yan, Zhulun Wang, Athena Sudom, Mario Cardozo, Michael DeGraffenreid, Marc Labelle

Bioorg Med Chem Lett· December 2010

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Identification of a PPARdelta agonist with partial agonistic activity on PPARgamma.
Richard V Connors, Zhulun Wang, Martin Harrison, Alex Zhang, Malgorzata Wanska, Marc Labelle

Bioorg Med Chem Lett· July 2009

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Synthesis and optimization of arylsulfonylpiperazines as a novel class of inhibitors of 11 beta-hydroxysteroid dehydrogenase type 1 (11 beta-HSD1).
Daqing Sun, Zhulun Wang, Mario Cardozo, Rebekah Choi, Michael Degraffenreid, Marc Labelle

Bioorg Med Chem Lett· March 2009

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Distinctive molecular inhibition mechanisms for selective inhibitors of human 11beta-hydroxysteroid dehydrogenase type 1.
Hua Tu, Jay P Powers, Jinsong Liu, Stefania Ursu, Athena Sudom, Marc Labelle

Bioorg Med Chem· October 2008

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Discovery and initial SAR of arylsulfonylpiperazine inhibitors of 11beta-hydroxysteroid dehydrogenase type 1 (11beta-HSD1).
Daqing Sun, Zhulun Wang, Yongmei Di, Juan C Jaen, Marc Labelle

Bioorg Med Chem Lett· June 2008

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Discovery of a potent and selective prostaglandin D2 receptor antagonist, [(3R)-4-(4-chloro-benzyl)-7-fluoro-5-(methylsulfonyl)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl]-acetic acid (MK-0524).
Claudio F Sturino, Gary O'Neill, Nicolas Lachance, Michael Boyd, Carl Berthelette, Marc Labelle

J Med Chem· February 2007

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Comparison between two classes of selective EP(3) antagonists and their biological activities.
Michel Belley, Chi Chung Chan, Yves Gareau, Michel Gallant, Hélène Juteau, Marc Labelle

Bioorg Med Chem Lett· November 2006

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Identification of an indole series of prostaglandin D2 receptor antagonists.
Claudio F Sturino, Nicolas Lachance, Michael Boyd, Carl Berthelette, Marc Labelle

Bioorg Med Chem Lett· June 2006

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Oxadiazole derivatives as a novel class of antimitotic agents: Synthesis, inhibition of tubulin polymerization, and activity in tumor cell lines.
Xiaohu Ouyang, Evgueni L Piatnitski, Vatee Pattaropong, Xiaoling Chen, Hai-Ying He, Marc Labelle

Bioorg Med Chem Lett· March 2006

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Pyrimido-oxazepine as a versatile template for the development of inhibitors of specific kinases.
Weitao Pan, Hu Liu, Yong-Jiang Xu, Xin Chen, Ki Hwan Kim, Marc Labelle

Bioorg Med Chem Lett· December 2005

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Synthesis and structure-activity relationships of 1,2,4-triazoles as a novel class of potent tubulin polymerization inhibitors.
Xiaohu Ouyang, Xiaoling Chen, Evgueni L Piatnitski, Alexander S Kiselyov, Hai-Ying He, Marc Labelle

Bioorg Med Chem Lett· December 2005

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Structure-activity relationship studies on ortho-substituted cinnamic acids, a new class of selective EP(3) antagonists.
Michel Belley, Michel Gallant, Bruno Roy, Karine Houde, Nicolas Lachance, Marc Labelle

Bioorg Med Chem Lett· February 2005

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Structure-activity relationship of triaryl propionic acid analogues on the human EP3 prostanoid receptor.
Michel Gallant, Michel Belley, Marie-Claude Carrière, Anne Chateauneuf, Danielle Denis, Marc Labelle

Bioorg Med Chem Lett· November 2003

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Liquid-Phase Synthesis with Solid-Phase Workup: Application to Multistep and Combinatorial Syntheses.
Hélène Perrier, Marc Labelle

J Org Chem· March 1999

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