Publications by authors named "Maria-Isabel Cadavid"

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Serotonin 2A receptor disulfide bridge integrity is crucial for ligand binding to different signalling states but not for its homodimerization.
Alba Iglesias, Marta Cimadevila, Rocío Ailim de la Fuente, María Martí-Solano, María Isabel Cadavid

Eur J Pharmacol· November 2017

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Targeting PDE10A GAF Domain with Small Molecules: A Way for Allosteric Modulation with Anti-Inflammatory Effects.
Ana M García, José Brea, Alejandro González-García, Concepción Pérez, María Isabel Cadavid

Molecules· September 2017

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Pharmacological tools based on imidazole scaffold proved the utility of PDE10A inhibitors for Parkinson's disease.
Ana M García, Irene G Salado, Daniel I Perez, José Brea, Jose A Morales-García, María Isabel Cadavid

Future Med Chem· May 2017

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Serotonin-2A homodimers are needed for signalling via both phospholipase A and phospholipase C in transfected CHO cells.
Alba Iglesias, Marta Cimadevila, María Isabel Cadavid, María Isabel Loza, José Brea

Eur J Pharmacol· April 2017

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Development of a Multiplex Assay for Studying Functional Selectivity of Human Serotonin 5-HT2A Receptors and Identification of Active Compounds by High-Throughput Screening.
Alba Iglesias, Sonia Lage, Maria Isabel Cadavid, Maria Isabel Loza, José Brea

J Biomol Screen· September 2016

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Modulation of cAMP-specific PDE without emetogenic activity: new sulfide-like PDE7 inhibitors.
Ana M García, José Brea, Jose A Morales-García, Daniel I Perez, Alejandro González, María Isabel Cadavid

J Med Chem· October 2014

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Unraveling phosphodiesterase surfaces. Identification of phosphodiesterase 7 allosteric modulation cavities.
Miriam Redondo, Ignacio Soteras, José Brea, Alejandro González-García, María Isabel Cadavid

Eur J Med Chem· September 2014

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The arylpiperazine derivatives N-(4-cyanophenylmethyl)-4-(2-diphenyl)-1-piperazinehexanamide and N-benzyl-4-(2-diphenyl)-1-piperazinehexanamide exert a long-lasting inhibition of human serotonin 5-HT7 receptor binding and cAMP signaling.
Patricio Atanes, Enza Lacivita, Javier Rodríguez, José Brea, Javier Burgueño, María Isabel Cadavid

Pharmacol Res Perspect· December 2013

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Synthesis and allosteric modulation of the dopamine receptor by peptide analogs of L-prolyl-L-leucyl-glycinamide (PLG) modified in the L-proline or L-proline and L-leucine scaffolds.
Joana Ferreira da Costa, Olga Caamaño, Franco Fernández, Xerardo García-Mera, Ivo E Sampaio-Dias, María Isabel Cadavid

Eur J Med Chem· November 2013

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Discovery of 3,4-Dihydropyrimidin-2(1H)-ones As a Novel Class of Potent and Selective A2B Adenosine Receptor Antagonists.
Abel Crespo, Abdelaziz El Maatougui, Pierfrancesco Biagini, Jhonny Azuaje, Alberto Coelho, María Isabel Cadavid

ACS Med Chem Lett· November 2013

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Selective and potent adenosine A3 receptor antagonists by methoxyaryl substitution on the N-(2,6-diarylpyrimidin-4-yl)acetamide scaffold.
Vicente Yaziji, David Rodríguez, Alberto Coelho, Xerardo García-Mera, Abdelaziz El Maatougui, María Isabel Cadavid

Eur J Med Chem· January 2013

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Identification in silico and experimental validation of novel phosphodiesterase 7 inhibitors with efficacy in experimental autoimmune encephalomyelitis mice.
Miriam Redondo, Valle Palomo, José Brea, Daniel I Pérez, Rocío Martín-Álvarez, María Isabel Cadavid

ACS Chem Neurosci· October 2012

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Effect of phosphodiesterase 7 (PDE7) inhibitors in experimental autoimmune encephalomyelitis mice. Discovery of a new chemically diverse family of compounds.
Miriam Redondo, José Brea, Daniel I Perez, Ignacio Soteras, Cristina Val, María Isabel Cadavid

J Med Chem· April 2012

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Discovery of LAS101057: A Potent, Selective, and Orally Efficacious A2B Adenosine Receptor Antagonist.
Paul Eastwood, Cristina Esteve, Jacob González, Silvia Fonquerna, Josep Aiguadé, María Isabel Cadavid

ACS Med Chem Lett· March 2011

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Pyrimidine derivatives as potent and selective A3 adenosine receptor antagonists.
Vicente Yaziji, David Rodríguez, Hugo Gutiérrez-de-Terán, Alberto Coelho, Olga Caamaño, María Isabel Cadavid

J Med Chem· January 2011

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Pyrazolo[1',5':1,6]pyrimido[4,5-d]pyridazin-4(3H)-ones as selective human A(1) adenosine receptor ligands.
Maria Paola Giovannoni, Claudia Vergelli, Agostino Cilibrizzi, Letizia Crocetti, Claudio Biancalani, Maria Isabel Cadavid

Bioorg Med Chem· November 2010

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Evidence for distinct antagonist-revealed functional states of 5-hydroxytryptamine(2A) receptor homodimers.
José Brea, Marián Castro, Jesús Giraldo, Juan F López-Giménez, Juan Fernando Padín, Maria Isabel Cadavid

Mol Pharmacol· June 2009

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Synthesis of novel 1-alkyl-8-substituted-3-(3-methoxypropyl) xanthines as putative A(2B) receptor antagonists.
María Isabel Nieto, María Carmen Balo, José Brea, Olga Caamaño, María Isabel Cadavid

Bioorg Med Chem· May 2009

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A new chemical tool (C0036E08) supports the role of adenosine A(2B) receptors in mediating human mast cell activation.
Montserrat Buceta, Eduardo Domínguez, Marián Castro, José Brea, David Alvarez, María Isabel Cadavid

Biochem Pharmacol· October 2008

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1-, 3- and 8-substituted-9-deazaxanthines as potent and selective antagonists at the human A2B adenosine receptor.
Angela Stefanachi, Jose Manuel Brea, Maria Isabel Cadavid, Nuria B Centeno, Cristina Esteve

Bioorg Med Chem· March 2008

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Synthesis, adenosine receptor binding and 3D-QSAR of 4-substituted 2-(2'-furyl)-1,2,4-triazolo[1,5-a]quinoxalines.
Ana Martínez, Hugo Gutiérrez-de-Terán, José Brea, Enrique Raviña, Maria Isabel Loza, Maria Isabel Cadavid

Bioorg Med Chem· February 2008

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Discovery and characterization of 4'-(2-furyl)-N-pyridin-3-yl-4,5'-bipyrimidin-2'-amine (LAS38096), a potent, selective, and efficacious A2B adenosine receptor antagonist.
Bernat Vidal, Arsenio Nueda, Cristina Esteve, Teresa Domenech, Sonia Benito, María Isabel Cadavid

J Med Chem· May 2007

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New pyrrolopyrimidin-6-yl benzenesulfonamides: potent A2B adenosine receptor antagonists.
Cristina Esteve, Arsenio Nueda, José Luis Díaz, Jorge Beleta, Alvaro Cárdenas, Maria Isabel Cadavid

Bioorg Med Chem Lett· July 2006

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Design, synthesis, and structure-activity relationships of 1-,3-,8-, and 9-substituted-9-deazaxanthines at the human A2B adenosine receptor.
Angelo Carotti, Maria Isabel Cadavid, Nuria B Centeno, Cristina Esteve, Maria Isabel Loza

J Med Chem· January 2006

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8-Substituted-9-deazaxanthines as adenosine receptor ligands: design, synthesis and structure-affinity relationships at A2B.
Angelo Carotti, Angela Stefanachi, Enrique Raviña, Eddy Sotelo, Maria Isabel Loza, Maria Isabel Cadavid

Eur J Med Chem· October 2004

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