Publications by authors named "Michele Matchett"

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Discovery of new indole-based acylsulfonamide Na1.7 inhibitors.
Yong-Jin Wu, Brian Venables, Jason Guernon, Jie Chen, Sing-Yuen Sit, Michele Matchett

Bioorg Med Chem Lett· February 2019

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Correction to Discovery of Indole- and Indazole-acylsulfonamides as Potent and Selective Na1.7 Inhibitors for the Treatment of Pain.
Guanglin Luo, Ling Chen, Amy Easton, Amy Newton, Clotilde Bourin, Michele Matchett

J Med Chem· February 2019

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Discovery of Indole- and Indazole-acylsulfonamides as Potent and Selective Na1.7 Inhibitors for the Treatment of Pain.
Guanglin Luo, Ling Chen, Amy Easton, Amy Newton, Clotilde Bourin, Michele Matchett

J Med Chem· January 2019

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Discovery of morpholine-based aryl sulfonamides as Na1.7 inhibitors.
Yong-Jin Wu, Jason Guernon, Andrea McClure, Brian Venables, Ramkumar Rajamani, Michele Matchett

Bioorg Med Chem Lett· March 2018

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Discovery of non-zwitterionic aryl sulfonamides as Na1.7 inhibitors with efficacy in preclinical behavioral models and translational measures of nociceptive neuron activation.
Yong-Jin Wu, Jason Guernon, Andrea McClure, Guanglin Luo, Ramkumar Rajamani, Michele Matchett

Bioorg Med Chem· October 2017

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Development of New Benzenesulfonamides As Potent and Selective Na1.7 Inhibitors for the Treatment of Pain.
Yong-Jin Wu, Jason Guernon, Jianliang Shi, Jonathan Ditta, Kevin J Robbins, Michele Matchett

J Med Chem· March 2017

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Design and Synthesis of a New Series of 4-Heteroarylamino-1'-azaspiro[oxazole-5,3'-bicyclo[2.2.2]octanes as α7 Nicotinic Receptor Agonists. 1. Development of Pharmacophore and Early Structure-Activity Relationship.
James Cook, F Christopher Zusi, Ivar M McDonald, Dalton King, Matthew D Hill, Michele Matchett

J Med Chem· December 2016

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Development of 1-Pyrazolo[3,4-]pyridines as Metabotropic Glutamate Receptor 5 Positive Allosteric Modulators.
Matthew D Hill, Haiquan Fang, Jeffrey M Brown, Thaddeus Molski, Amy Easton, Michele Matchett

ACS Med Chem Lett· December 2016

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Oxazolidinone-based allosteric modulators of mGluR5: Defining molecular switches to create a pharmacological tool box.
Hong Huang, Andrew P Degnan, Anand Balakrishnan, Amy Easton, Michael Gulianello, Michele Matchett

Bioorg Med Chem Lett· September 2016

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Discovery and Preclinical Evaluation of BMS-955829, a Potent Positive Allosteric Modulator of mGluR5.
Fukang Yang, Lawrence B Snyder, Anand Balakrishnan, Jeffrey M Brown, Digavalli V Sivarao, Michele Matchett

ACS Med Chem Lett· March 2016

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Evaluation and optimization of compound solubilization and delivery methods in a two-tiered ion channel lead optimization triage.
Adam W Hendricson, Liz Gallagher, Michele Matchett, Meredith Ferrante, Steve Spence

Assay Drug Dev Technol· April 2012

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Design of an automated enhanced-throughput platform for functional characterization of positive allosteric modulator-induced leftward shifts in apparent agonist potency in vitro.
Adam Hendricson, Michele Matchett, Meredith Ferrante, Chris Ferrante, Ed Hunnicutt

J Lab Autom· April 2012

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Characterization of N-(adamantan-1-ylmethyl)-5-[(3R-amino-pyrrolidin-1-yl)methyl]-2-chloro-benzamide, a P2X7 antagonist in animal models of pain and inflammation.
Daniel C Broom, David J Matson, Elizabeth Bradshaw, Marianne E Buck, Robin Meade, Michele Matchett

J Pharmacol Exp Ther· December 2008

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The P2X3 antagonist P1, P5-di[inosine-5'] pentaphosphate binds to the desensitized state of the receptor in rat dorsal root ganglion neurons.
Kristen K Ford, Michele Matchett, James E Krause, Weifeng Yu

J Pharmacol Exp Ther· October 2005

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