Publications by authors named "Randal Bugianesi"

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Design, synthesis and biological evaluation of indane derived GPR40 agoPAMs.
Barbara Pio, Harry R Chobanian, Yan Guo, Hubert Josien, William K Hagmann, Randal Bugianesi

Bioorg Med Chem Lett· July 2019

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Design and Synthesis of Novel, Selective GPR40 AgoPAMs.
Christopher W Plummer, Matthew J Clements, Helen Chen, Murali Rajagopalan, Hubert Josien, Randal Bugianesi

ACS Med Chem Lett· February 2017

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Discovery and Optimization of a Novel Triazole Series of GPR142 Agonists for the Treatment of Type 2 Diabetes.
Liangqin Guo, Dann L Parker, Yi Zang, Ramzi F Sweis, Weiguo Liu, Randal Bugianesi

ACS Med Chem Lett· December 2016

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Discovery and development of benzo-[1,2,4]-triazolo-[1,4]-oxazepine GPR142 agonists for the treatment of diabetes.
Jonathan E Wilson, Ravi Kurukulasuriya, Christopher Sinz, Matthew Lombardo, Kate Bender, Randal Bugianesi

Bioorg Med Chem Lett· June 2016

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Definitive Metabolite Identification Coupled with Automated Ligand Identification System (ALIS) Technology: A Novel Approach to Uncover Structure-Activity Relationships and Guide Drug Design in a Factor IXa Inhibitor Program.
Ting Zhang, Yong Liu, Xianshu Yang, Gary E Martin, Huifang Yao, Randal M Bugianesi

J Med Chem· March 2016

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Improved Cav2.2 Channel Inhibitors through a gem-Dimethylsulfone Bioisostere Replacement of a Labile Sulfonamide.
Pengcheng P Shao, Feng Ye, Prasun K Chakravarty, James B Herrington, Ge Dai, Randal M Bugianesi

ACS Med Chem Lett· November 2013

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Aminopiperidine sulfonamide Cav2.2 channel inhibitors for the treatment of chronic pain.
Pengcheng P Shao, Feng Ye, Prasun K Chakravarty, Deepu J Varughese, James B Herrington, Randal M Bugianesi

J Med Chem· November 2012

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Characterization of the substituted N-triazole oxindole TROX-1, a small-molecule, state-dependent inhibitor of Ca(V)2 calcium channels.
Andrew M Swensen, James Herrington, Randal M Bugianesi, Ge Dai, Rodolfo J Haedo

Mol Pharmacol· March 2012

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Analgesic effects of a substituted N-triazole oxindole (TROX-1), a state-dependent, voltage-gated calcium channel 2 blocker.
Catherine Abbadie, Owen B McManus, Shu-Yu Sun, Randal M Bugianesi, Ge Dai

J Pharmacol Exp Ther· August 2010

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A high-throughput assay for evaluating state dependence and subtype selectivity of Cav2 calcium channel inhibitors.
Ge Dai, Rodolfo J Haedo, Vivien A Warren, Kevin S Ratliff, Randal M Bugianesi

Assay Drug Dev Technol· April 2008

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Blockers of the delayed-rectifier potassium current in pancreatic beta-cells enhance glucose-dependent insulin secretion.
James Herrington, Yun-Ping Zhou, Randal M Bugianesi, Paula M Dulski, Yue Feng

Diabetes· April 2006

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A cell-sparing electric field stimulation technique for high-throughput screening of voltage-gated ion channels.
Randal M Bugianesi, Paul R Augustine, Karim Azer, Claude Dufresne, James Herrington

Assay Drug Dev Technol· February 2006

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A high-capacity membrane potential FRET-based assay for NaV1.8 channels.
Chou J Liu, Birgit T Priest, Randal M Bugianesi, Paula M Dulski, John P Felix

Assay Drug Dev Technol· February 2006

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B
Biophysical and pharmacological properties of the voltage-gated potassium current of human pancreatic beta-cells.
James Herrington, Manuel Sanchez, Denize Wunderler, Lizhen Yan, Randal M Bugianesi

J Physiol· August 2005

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Stichodactyla helianthus peptide, a pharmacological tool for studying Kv3.2 channels.
Lizhen Yan, James Herrington, Ethan Goldberg, Paula M Dulski, Randal M Bugianesi

Mol Pharmacol· May 2005

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Potent Kv1.3 inhibitors from correolide-modification of the C18 position.
Jianming Bao, Shouwu Miao, Frank Kayser, Andrew J Kotliar, Robert K Baker, Randal M Bugianesi

Bioorg Med Chem Lett· January 2005

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Expression of voltage-gated potassium channels in human and rhesus pancreatic islets.
Lizhen Yan, David J Figueroa, Christopher P Austin, Yuan Liu, Randal M Bugianesi

Diabetes· March 2004

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Substitution of a single residue in Stichodactyla helianthus peptide, ShK-Dap22, reveals a novel pharmacological profile.
Richard E Middleton, Manuel Sanchez, Ana-Rosa Linde, Randal M Bugianesi, Ge Dai

Biochemistry· November 2003

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Identification of a new class of inhibitors of the voltage-gated potassium channel, Kv1.3, with immunosuppressant properties.
William A Schmalhofer, Jianming Bao, Owen B McManus, Brian Green, Mary Matyskiela, Randal M Bugianesi

Biochemistry· June 2002

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