Publications by authors named "Simon Gaines"

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From PIM1 to PI3Kδ via GSK3β: Target Hopping through the Kinome.
Zoë A Henley, Benjamin D Bax, Laura M Inglesby, Aurélie Champigny, Simon Gaines

ACS Med Chem Lett· October 2017

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Palladium-Catalyzed Ring Expansion of Spirocyclopropanes to Form Caprolactams and Azepanes.
Olivier René, Iain A Stepek, Alberto Gobbi, Benjamin P Fauber, Simon Gaines

J Org Chem· October 2015

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A reversed sulfonamide series of selective RORc inverse agonists.
Monique B van Niel, Benjamin P Fauber, Matthew Cartwright, Simon Gaines, Jonathan C Killen

Bioorg Med Chem Lett· December 2014

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Identification of C-2 hydroxyethyl imidazopyrrolopyridines as potent JAK1 inhibitors with favorable physicochemical properties and high selectivity over JAK2.
Mark Zak, Christopher A Hurley, Stuart I Ward, Philippe Bergeron, Kathy Barrett, Simon Gaines

J Med Chem· June 2013

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Irreversible 4-Aminopiperidine Transglutaminase 2 Inhibitors for Huntington's Disease.
Michael E Prime, Frederick A Brookfield, Stephen M Courtney, Simon Gaines, Richard W Marston

ACS Med Chem Lett· September 2012

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The characterization of a novel V1b antagonist lead series.
Chris A Smethurst, Jennifer A Borthwick, Simon Gaines, Steve Watson, Andrew Green

Bioorg Med Chem Lett· January 2011

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Identification of a sulfonamide series of CCR2 antagonists.
Simon Peace, Joanne Philp, Carl Brooks, Val Piercy, Kitty Moores, Simon Gaines

Bioorg Med Chem Lett· July 2010

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The identification of beta-hydroxy carboxylic acids as selective MMP-12 inhibitors.
Ian P Holmes, Simon Gaines, Steve P Watson, Olivier Lorthioir, Adam Walker

Bioorg Med Chem Lett· October 2009

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Dopamine D3 receptor antagonists: the quest for a potentially selective PET ligand. Part one: lead identification.
Ian P Holmes, Fabrizio Micheli, Simon Gaines, Olivier Lorthioir, Steve P Watson

Bioorg Med Chem Lett· August 2009

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Large Molecular Quadratic Hyperpolarizabilities in Donor/Acceptor-Substituted trans-Tetraammineruthenium(II) Complexes.
Benjamin J. Coe, Michelle C. Chamberlain, Jonathan P. Essex-Lopresti, Simon Gaines, John C. Jeffery

Inorg Chem· July 1997

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