Publications by authors named "Gavin Collie"

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Use of Direct-to-Biology Strategies for the Discovery of 2'-Deoxynucleoside 5'-Monophosphate N-Glycosidase (DNPH1) PROTACs.
Niall A Anderson, Bernard Barlaam, Argyrides Argyrou, Peter C Astles, Hanna Bruss, Gavin W Collie

J Med Chem· November 2025

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Discovery and Optimization of a Non-Nucleoside-Based Series of Inhibitors of 2'-Deoxynucleoside 5'-Monophosphate Glycosidase (DNPH1).
Bernard Barlaam, Luz Alonso-Crisostomo, Niall A Anderson, Argyrides Argyrou, Peter C Astles, Gavin W Collie

J Med Chem· November 2025

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Focused Structure-Based Virtual Screening Identifies Novel Inhibitors of SOS1.
Silvia Bonomo, Floriane Gibault, Sharan K Bagal, J Henry Blackwell, Jason Breed, Gavin W Collie

ACS Med Chem Lett· October 2025

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Discovery of AZD8421: A Potent CDK2 Inhibitor with Selectivity Against Other CDK Family Members and the Human Kinome.
Avipsa Ghosh, Afshan Ahmed, Konstantina Amoiradaki, Amber Y S Balazs, Bernard Barlaam, Gavin W Collie

J Med Chem· September 2025

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Structural and Molecular Insight into the PWWP1 Domain of NSD2 from the Discovery of Novel Binders Via DNA-Encoded Library Screening.
Gavin W Collie, Bryony Ackroyd, Catriona Corbishley, Daniel H O'Donovan, Alex Edwards

ACS Med Chem Lett· September 2025

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Discovery of a Series of Covalent Ligands That Bind to Cys77 of the Von Hippel-Lindau Tumor Suppressor Protein (VHL).
Simon C C Lucas, Yong Xu, Sarah Hewitt, Gavin W Collie, Lucia Fusani

ACS Med Chem Lett· April 2025

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Guanidinium-Stapled Helical Peptides for Targeting Protein-Protein Interactions.
Camille Perdriau, Anaïs Luton, Katharina Zimmeter, Maxime Neuville, Claire Saragaglia, Gavin W Collie

Angew Chem Int Ed Engl· January 2025

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Specific radiation damage to halogenated inhibitors and ligands in protein-ligand crystal structures.
Matthew J Rodrigues, Marc Cabry, Gavin Collie, Michael Carter, Craig McAndrew

J Appl Crystallogr· December 2024

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Innovative Self-Assembly of 15-Mer Chimeric α-Peptide-Oligourea Foldamers toward Cl-Selective Ion Channels.
Chiranjit Dutta, Pannaga Krishnamurthy, Dandan Su, Jianwei Li, Sung Hyun Yoo, Gavin W Collie

Small Sci· August 2024

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Fragment-Based Discovery of Novel MUS81 Inhibitors.
Gavin W Collie, Ulf Börjesson, Yunhua Chen, Zhiqiang Dong, Paolo Di Fruscia

ACS Med Chem Lett· July 2024

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Identification of Novel Potent NSD2-PWWP1 Ligands Using Structure-Based Design and Computational Approaches.
Luca Carlino, Peter C Astles, Bryony Ackroyd, Afshan Ahmed, Christina Chan, Gavin W Collie

J Med Chem· June 2024

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Oligourea helix bundle binds detergents with diverse polar head groups.
Sung Hyun Yoo, Jérémie Buratto, Arup Roy, Morgane Pasco, Karolina Pulka-Ziach, Gavin W Collie

Org Biomol Chem· January 2024

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Screening Ultra-Large Encoded Compound Libraries Leads to Novel Protein-Ligand Interactions and High Selectivity.
Gavin W Collie, Matthew A Clark, Anthony D Keefe, Andrew Madin, Jon A Read

J Med Chem· January 2024

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Correction to "E3 Ligases Meet Their Match: Fragment-Based Approaches to Discover New E3 Ligands and to Unravel E3 Biology".
Iacovos N Michaelides, Gavin W Collie

J Med Chem· November 2023

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Discovery and Optimization of the First ATP Competitive Type-III c-MET Inhibitor.
Iacovos N Michaelides, Gavin W Collie, Ulf Börjesson, Christina Vasalou, Omar Alkhatib

J Med Chem· July 2023

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E3 Ligases Meet Their Match: Fragment-Based Approaches to Discover New E3 Ligands and to Unravel E3 Biology.
Iacovos N Michaelides, Gavin W Collie

J Med Chem· March 2023

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Discovery of a selective c-MET inhibitor with a novel binding mode.
Gavin W Collie, Louise Barlind, Sana Bazzaz, Ulf Börjesson, Ian L Dale

Bioorg Med Chem Lett· November 2022

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Discovering cell-active BCL6 inhibitors: effectively combining biochemical HTS with multiple biophysical techniques, X-ray crystallography and cell-based assays.
Olivier A Pierrat, Manjuan Liu, Gavin W Collie, Kartika Shetty, Matthew J Rodrigues

Sci Rep· November 2022

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Adaptive Binding of Alkyl Glycosides by Nonpeptidic Helix Bundles in Water: Toward Artificial Glycolipid Binding Proteins.
Sung Hyun Yoo, Jérémie Buratto, Arup Roy, Estelle Morvan, Morgane Pasco, Gavin W Collie

J Am Chem Soc· September 2022

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Racemic crystal structures of A-DNA duplexes.
Pradeep K Mandal, Gavin W Collie, Brice Kauffmann, Ivan Huc

Acta Crystallogr D Struct Biol· June 2022

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Optimizing Shape Complementarity Enables the Discovery of Potent Tricyclic BCL6 Inhibitors.
Owen A Davis, Kwai-Ming J Cheung, Alfie Brennan, Matthew G Lloyd, Matthew J Rodrigues, Gavin W Collie

J Med Chem· June 2022

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Into Deep Water: Optimizing BCL6 Inhibitors by Growing into a Solvated Pocket.
Matthew G Lloyd, Rosemary Huckvale, Kwai-Ming J Cheung, Matthew J Rodrigues, Gavin W Collie

J Med Chem· December 2021

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Crystal structures capture multiple stoichiometric states of an aqueous self-assembling oligourea foldamer.
Gavin W Collie, Caterina M Lombardo, Sung Hyun Yoo, Karolina Pułka-Ziach, Valérie Gabelica

Chem Commun (Camb)· September 2021

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Fragment-Based Discovery of Novel Allosteric MEK1 Binders.
Paolo Di Fruscia, Fredrik Edfeldt, Igor Shamovsky, Gavin W Collie, Anna Aagaard

ACS Med Chem Lett· February 2021

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Structural Basis for Targeting the Folded P-Loop Conformation of c-MET.
Gavin W Collie, Iacovos N Michaelides, Kevin Embrey, Christopher J Stubbs, Ulf Börjesson

ACS Med Chem Lett· January 2021

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