Publications by authors named "Helmut Buschmann"

Claim this Profile
M
Mechanochemical Degradation of Active Pharmaceutical Ingredients (APIs): A Simple Tool for the Prediction of Drug Stability.
Ulrike Holzgrabe, Helmut Buschmann, Norbert Handler, Mostafa M Amer, Renè Hommelsheim

Chimia (Aarau)· September 2025

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
T
The conserved core nuclear egress complex (NEC) as an antiherpesviral drug target: Pharmacophore-based identification of NEC-specific inhibitors.
Julia Tillmanns, Verena Battisti, Jintawee Kicuntod, Friedrich Hahn, Debora Obergfäll, Helmut Buschmann

Antiviral Res· July 2025

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
D
Discovery of AIC263282, a Hepatitis B Virus Capsid Assembly Modulator Ready for Candidate Profiling.
Bernhard Lesch, Alexander Birkmann, Susanne Bonsmann, Alastair Donald, Florian Engel, Helmut Buschmann

J Med Chem· March 2025

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
P
Prediction of Degradation Profiles for Various Sartans under Solvent-Free Mechanochemical Conditions.
Mostafa M Amer, Laura Backer, Helmut Buschmann, Norbert Handler, Oliver Scherf-Clavel

Anal Chem· August 2024

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
A
Application of advanced high resolution mass spectrometric techniques for the analysis of losartan potassium regarding known and unknown impurities.
Laura Backer, Helmut Buschmann, Martina Kinzig, Fritz Sörgel, Oliver Scherf-Clavel

J Pharm Biomed Anal· March 2024

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
T
The quality of drugs and drug products - Always guaranteed?
Helmut Buschmann, Norbert Handler, Ulrike Holzgrabe

J Pharm Biomed Anal· February 2024

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
S
Structure-based Design of Novel Hepatitis B Virus Capsid Assembly Modulators.
Elena Detta, Angelica Corcuera, Andreas Urban, Thomas Goldner, Susanne Bonsmann, Helmut Buschmann

Bioorg Med Chem Lett· September 2023

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
M
Mechanochemical Oxidative Degradation of Thienopyridine Containing Drugs: Toward a Simple Tool for the Prediction of Drug Stability.
Everaldo F Krake, Laura Backer, Benjamin Andres, Wolfgang Baumann, Norbert Handler, Helmut Buschmann

ACS Cent Sci· June 2023

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
D
Discovery, Chemistry, and Preclinical Development of Pritelivir, a Novel Treatment Option for Acyclovir-Resistant Herpes Simplex Virus Infections.
Alexander Birkmann, Susanne Bonsmann, Dirk Kropeit, Tamara Pfaff, Manickam Rangaraju, Helmut Buschmann

J Med Chem· October 2022

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
A
An automated microfluidic platform for the screening and characterization of novel hepatitis B virus capsid assembly modulators.
Tamás Vermes, Mark Kielpinski, Thomas Henkel, Miquel A Pericàs, Esther Alza, Helmut Buschmann

Anal Methods· January 2022

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
B
Ball milling - a new concept for predicting degradation profiles in active pharmaceutical ingredients.
Reinhard P Kaiser, Everaldo F Krake, Laura Backer, Jonas Urlaub, Wolfgang Baumann, Helmut Buschmann

Chem Commun (Camb)· November 2021

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
D
Different solid forms for optimizing route of administration of the herpes drug Pritelivir.
Helga Ruebsamen-Schaeff, Helmut Buschmann

Medchemcomm· November 2019

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
D
Diffusion ordered NMR spectroscopy measurements as screening method of potential reactions of API and excipients in drug formulations.
Alexander Becht, Curd Schollmayer, Johannes Wiest, Detlef Heller, Wolfgang Baumann, Helmut Buschmann

J Pharm Biomed Anal· January 2019

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
L
Lead Development of Thiazolylsulfonamides with Carbonic Anhydrase Inhibitory Action.
Fabrizio Carta, Alexander Birkmann, Tamara Pfaff, Helmut Buschmann, Wilfried Schwab

J Med Chem· April 2017

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
N
New approaches to treating pain.
Andrea Wolkerstorfer, Norbert Handler, Helmut Buschmann

Bioorg Med Chem Lett· February 2016

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
A
An RNA Hybridization Assay for Screening Influenza A Virus Polymerase Inhibitors Using the Entire Ribonucleoprotein Complex.
Franz-Ferdinand Roch, Georg Hinterkörner, John Menke, Guo-Qing Tang, Stephen Cusack, Helmut Buschmann

Assay Drug Dev Technol· October 2015

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
S
Sigma-1 receptor antagonism as opioid adjuvant strategy: enhancement of opioid antinociception without increasing adverse effects.
Alba Vidal-Torres, Beatriz de la Puente, Maria Rocasalbas, Clara Touriño, Simona Andreea Bura, Helmut Buschmann

Eur J Pharmacol· July 2013

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
N
N-cyano sulfoximines: COX inhibition, anticancer activity, cellular toxicity, and mutagenicity.
Seong Jun Park, Hannah Baars, Stefanie Mersmann, Helmut Buschmann, Jens Malte Baron

ChemMedChem· February 2013

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
S
Synthesis and biological evaluation of the 1-arylpyrazole class of σ(1) receptor antagonists: identification of 4-{2-[5-methyl-1-(naphthalen-2-yl)-1H-pyrazol-3-yloxy]ethyl}morpholine (S1RA, E-52862).
José Luis Díaz, Rosa Cuberes, Joana Berrocal, Montserrat Contijoch, Ute Christmann, Helmut Buschmann

J Med Chem· October 2012

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
M
Microwave assisted synthesis of spirocyclic pyrrolidines -σ1 receptor ligands with modified benzene-N-distance.
Annemarie Jasper, Dirk Schepmann, Kirstin Lehmkuhl, Jose Miguel Vela, Helmut Buschmann

Eur J Med Chem· July 2012

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
S
Syntheses and biological activities of sulfoximine-based acyclic triaryl olefins.
Xiao Yun Chen, Seong Jun Park, Helmut Buschmann, Maria De Rosa, Carsten Bolm

Bioorg Med Chem Lett· July 2012

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
M
Mechanistic and functional differentiation of tapentadol and tramadol.
Robert B Raffa, Helmut Buschmann, Thomas Christoph, Gary Eichenbaum, Werner Englberger

Expert Opin Pharmacother· July 2012

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
T
Thiophene bioisosteres of spirocyclic σ receptor ligands: relationships between substitution pattern and σ receptor affinity.
Christoph Oberdorf, Dirk Schepmann, Jose Miguel Vela, Helmut Buschmann, Jörg Holenz

J Med Chem· June 2012

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
C
Combination of two pharmacophoric systems: synthesis and pharmacological evaluation of spirocyclic pyranopyrazoles with high σ₁ receptor affinity.
Torsten Schläger, Dirk Schepmann, Kirstin Lehmkuhl, Jörg Holenz, Jose Miguel Vela, Helmut Buschmann

J Med Chem· October 2011

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
B
Bioactive sulfoximines: syntheses and properties of Vioxx analogs.
Seong Jun Park, Helmut Buschmann, Carsten Bolm

Bioorg Med Chem Lett· August 2011

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis